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(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[2-(4H-1,2,4-triazol-4-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylic acid
N-[2-methyl-1-(pyridin-3-yl)propyl]-4-pentanamidobenzamide
2,3-dimethoxy-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
1-(4-chlorophenyl)-N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]cyclopropane-1-carboxamide
(3S,4R)-N,N-dimethyl-1-(2-methyl-1-benzofuran-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
N-[3-(2-methoxyethoxy)phenyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-hydroxy-N-propyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}-4-phenylbenzamide
2-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(1H-pyrazol-1-yl)acetamide
N-methyl-4-{1-[2-(pyridin-4-yl)ethyl]-1H-imidazol-2-yl}benzene-1-sulfonamide
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol
N4-[(2,5-difluorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[2-(hydroxymethyl)piperidin-1-yl]pyridine-3-carboxamide
4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3λ6,4-oxathiazinane-3,3-dione
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]pyridine-3-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
[(1-{[1-(3,5-dimethylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
(3R,4R)-3-cyclopropyl-4-methyl-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
2-(3-methoxypropyl)-8-[2-oxo-2-(piperazin-1-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
N3-cyclopentyl-1-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-(2-fluorophenoxymethyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-ethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}ethan-1-one
2-butoxy-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-cyclopentyl-4-[(3,5-dichloropyridin-4-yl)methyl]-1,4-diazepane
2,4-dimethyl-N-[4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)phenyl]benzamide
2-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
3-(2-methylpropyl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1,2-oxazole-5-carboxamide
N-(3-{methyl[(3-methylpyridin-4-yl)methyl]carbamoyl}phenyl)oxolane-2-carboxamide
4-benzyl-N-(3-acetamidophenyl)-4-hydroxypiperidine-1-carboxamide
N,1-dimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
4-{2-[1-(4-methylpiperazine-1-carbonyl)piperidin-2-yl]ethyl}phenol
1-[(3S,4R)-1-(5-chloro-2-methoxybenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
(2E)-1-[4-(butylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
2-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)-1,2-oxazinane
2-{2-[4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
methyl 2-{[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazol-7-yl]formamido}-4-(methylsulfanyl)butanoate
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
N-{2-[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-[4-(furan-2-ylmethoxy)phenyl]-3-propoxypiperidine-1-carboxamide
N-methyl-N-[2-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)ethyl]-2-phenylbutanamide
5-(2-benzylpropanoyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxypyridine-4-carboxamide
N-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(5S,9aS,9bS)-2-cyclopentyl-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-3-(1-methylpiperidin-4-yl)propanamide