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{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
5-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-N-phenylpyrimidin-2-amine
(2R,3R)-3-amino-1'-[2-(ethylamino)pyrimidine-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-(2-chlorophenyl)-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methylfuran-2-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylacetamide
7-methyl-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-ethyl-N-[4-(pyridin-2-yl)butyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[4-(propan-2-yl)phenyl]-1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-amine
N-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-2-(pyrrolidin-3-yl)benzamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-1-[(4-ethynylphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-{5-[(2-phenyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
6-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-fluoro-N,2-dimethyl-N-[1-(pyridin-3-yl)pentyl]quinoline-4-carboxamide
5-(3-chloro-4-methoxybenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
2-methoxy-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-3-carbonitrile
N-[3-({[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
(2S)-3-(4-hydroxyphenyl)-2-{[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]formamido}propanamide
(1S,5R)-6-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(1-cyclohexyl-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
6-methyl-1-(3-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}propyl)-1,2-dihydropyridin-2-one
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(furan-2-ylmethyl)propanamide
3-[(dimethylamino)methyl]-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidin-3-ol
4-({[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
(2E)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-3-(pyridin-2-yl)prop-2-enamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[3-(2-phenylpyridin-4-yl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
(3aR,5R,6S,7aS)-2-{[3-(trifluoromethyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
7-(2-methylphenyl)-4-(piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[5-(3-cyclopropyl-1H-pyrazol-5-yl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(2S)-1-({3-[4-(4-fluorophenyl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)pyrrolidine-2-carboxamide
6-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
5-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyridin-2-amine
4-(5-fluoro-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)morpholine
2-(furan-2-yl)-N-[(1-methylpiperidin-3-yl)methyl]-2-oxoacetamide
(3S,4R)-4-phenyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-cyclopropyl-4-methoxy-2-[(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)oxy]benzamide
2-[2-(3-acetylpiperidin-1-yl)-2-oxoethyl]-2-azaspiro[4.5]decan-3-one
1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
1-(3-methoxy-4-{[3-(thiomorpholine-4-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
4-methoxy-N-(2-methoxyethyl)-2-({1-[1-(1-methylcyclopropyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
(1R,5S,6R,7S)-3-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-{[(1-acetylpiperidin-4-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxo-N-phenylacetamide
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(1-methylcyclopropyl)propan-1-one
5-(3-propyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
3-[(3R,4S)-1-(5-methyl-1H-indazole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol