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(1R,3S,5S)-8-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
2,5-dimethyl-3-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrazine
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}benzamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
3-(4-fluorophenyl)-4-(5-methoxy-3-methyl-1H-indole-2-carbonyl)piperazin-2-one
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-4-phenyl-1,2,3,6-tetrahydropyridine-1-carboxamide
(1R,3S)-3-{[3-(4-methylbenzenesulfonamido)propyl]carbamoyl}cyclopentane-1-carboxylic acid
N-[5-({[2-(dimethylamino)-2-(3-methylphenyl)ethyl]carbamoyl}amino)-2-fluorophenyl]acetamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
2-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-4-carbonitrile
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-3-propylurea
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
(3R,4S)-1-(1-benzofuran-5-carbonyl)-3,4-dimethylpiperidin-4-ol
N-(propan-2-yl)-2-(4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperazin-1-yl)pyridine-4-carboxamide
3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-1-(prop-2-en-1-yl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
{[(3S,4R)-1-(2-chloro-5-fluorobenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(4-fluorophenyl)-2-hydroxyethan-1-one
N-[(4-methyl-1H-imidazol-5-yl)methyl]-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-amine
(4S)-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-({1-[(1R,2S)-2-(4-methylbenzoyl)cyclohexanecarbonyl]piperidin-4-yl}methyl)acetamide
N-[4-(1H-imidazol-1-yl)phenyl]-4-(morpholine-4-carbonyl)piperidine-1-carboxamide
(1R,5S)-N-(6-fluoropyridin-3-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(2-{4-[2-(trifluoromethyl)morpholine-4-carbonyl]phenoxy}ethyl)acetamide
9-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-(3,5-dimethyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanamide
N-ethyl-N-methyl-3-{[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]sulfamoyl}benzamide
7-chloro-3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]methyl}-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
3-[(methylsulfanyl)methyl]-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(1H-pyrazol-3-ylmethyl)amine
N-methyl-N-propyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
1-[4-(hydroxymethyl)benzoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-({[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
(2S,4R)-4-amino-1-[(4-ethylpiperazin-1-yl)sulfonyl]-N-methylpyrrolidine-2-carboxamide
8-(2,2-dimethylpropyl)-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4S)-1-(2-amino-2-methylpropyl)-3,3,4-trimethylpiperidin-4-ol
3-[1-(2-aminopyridine-4-carbonyl)piperidin-4-yl]-4-benzyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3R,4S)-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-{4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}pyridine
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
1-[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl]piperidine-4-carbonitrile
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-propyl-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4,4,4-trifluoro-N-[(3R,4S)-1-(3-hydroxypropyl)-4-(propan-2-yl)pyrrolidin-3-yl]butanamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][3-(dimethylamino)-2,2-dimethylpropyl]methylamine
{[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amine
2,6-dimethyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)quinoline-4-carboxamide