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2-cyclopropyl-4-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-(5-methylfuran-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-5-carboxamide
1-{[4-(furan-2-yl)phenyl]methyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-[(2R,3R,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,5,6-trimethylpyrimidin-4-amine
1-[4-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
N-(5-{[({1-[ethyl(methyl)amino]cyclohexyl}methyl)carbamoyl]amino}-2-methoxyphenyl)acetamide
3-[({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
2-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(5-methanesulfonyl-2-methylphenyl)-1-[3-(4-methoxyphenyl)propyl]urea
4-phenoxy-1-(3-phenylbutyl)piperidine-4-carboxylic acid
4-cyclobutyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,6-dimethylpyrimidin-2-amine
{4-[(4-methoxyphenyl)methyl]-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl}methanol
1-[1-(3,5-difluorophenyl)ethyl]-3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
[1-(2-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)piperidin-3-yl]methanol
8-[(2R)-2-hydroxypropanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methanesulfonamide
N-methyl-6-[(6-methylpyridin-2-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({1-[2-(trifluoromethyl)phenyl]ethyl})amine
4-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,6-dimethylpyrimidine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(prop-2-en-1-yl)-1H-pyrazole
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-{5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
3-(2,5-dioxoimidazolidin-4-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]propanamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N4-{1-oxaspiro[4.5]decan-3-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(2S,4S)-4-amino-N-methyl-1-[2-(4-phenylpiperidin-1-yl)acetyl]pyrrolidine-2-carboxamide
2-(thiomorpholin-4-yl)-2-[3-(2,2,2-trifluoroethoxy)phenyl]acetic acid
3-{[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]methyl}benzoic acid
2-[3-(3-methoxypropyl)piperidine-1-carbonyl]-6-methylphenol
(2R)-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}oxolane-2-carboxamide
2-chloro-4-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
5-{[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-methylfuran-2-carboxamide
4-hydroxy-N-[2-(methylsulfamoyl)ethyl]-2-phenylpyrimidine-5-carboxamide
4-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
1-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}azocane
(3R,4S)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-propylpyrrolidin-3-amine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-(1H-pyrazol-1-yl)butanamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(ethoxymethyl)piperidine
N-[(2S,4R,6S)-2-benzyl-6-(6-methoxypyridin-3-yl)oxan-4-yl]acetamide
methyl (2S,4R)-4-(2,2-diphenylacetamido)-1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
ethyl 1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
4-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
N3-(1H-1,3-benzodiazol-2-ylmethyl)-N5-butyl-1-cyclohexyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3S,4R)-1-(isoquinolin-1-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
{4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-3-(hydroxymethyl)phenyl}methanol
2-[(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]pyridine-4-carbonitrile
1-methyl-N-(2-phenylethyl)-5-[(propan-2-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide