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2-{[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-propylpyrrolidin-3-yl]amino}pyridine-3-carboxamide
3-benzoyl-1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
5-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-cyclopropylpyrrolidin-2-one
1-{[2-(difluoromethoxy)phenyl]methyl}-4-(2-phenoxyethyl)piperazine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(2-methylpropyl)-1,3-oxazole-4-carboxamide
2-(4-{[3-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
(2S,4S,5R)-5-(3-chlorophenyl)-4-[(3-hydroxypropyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-methyl-1,3-benzoxazole-6-carboxamide
1-[(2,5-dichlorophenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
2-(4-chloro-2-methylphenoxy)-1-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(5-methylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
4-{[2-(dimethylamino)ethyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
(2S,4R)-4-amino-1-(naphthalene-1-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)-2-methylheptan-2-ol
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyrazin-2-ylmethyl)propanamide
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(1H-pyrazol-1-yl)butan-1-one
2-(azocane-1-carbonyl)-5-fluoro-1,3-dimethyl-1H-indole
ethyl 1-[(2-methoxyphenyl)carbamoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-(3-phenylpropyl)piperidin-3-yl)methanol
6-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}acetamide
1-[(1R,5R)-6-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-methyl-2-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)-3,4-dihydropyrimidin-4-one
(1R,5S)-8-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
N-(3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)methanesulfonamide
3-{6-amino-5-cyano-4-[2-(furan-2-yl)phenyl]pyridin-2-yl}-1H-pyrazole-5-carboxylic acid
(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-({[2-(diethylamino)-2-(furan-2-yl)ethyl]amino}methyl)phenol
2-chloro-5-acetamido-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
6,7-dimethyl-4-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}-2H-chromen-2-one
methyl 6-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyridine-3-carboxylate
2-(4-ethylpiperazin-1-yl)-N-[1-(pyridin-3-yl)propan-2-yl]-2,3-dihydro-1H-indene-2-carboxamide
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propanamide
2-amino-6-(4-hydroxyphenyl)-5-methyl-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-6-ethyl-2-methylquinoline-4-carboxamide
1,4-dimethyl-9-[3-(1H-pyrazol-4-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
N-(1H-1,2,4-triazol-3-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-[5-(5-ethyl-1,3-oxazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(2-hydroxyethyl)propanamide
N-[(3S,4R)-4-(propan-2-yl)-1-(quinolin-4-yl)pyrrolidin-3-yl]acetamide
(2S,4R)-4-amino-N-ethyl-1-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]pyrrolidine-2-carboxamide
N-[2-(dimethylamino)ethyl]-3-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propanamide
7-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N4-(oxolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-(morpholine-4-carbonyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-(1H-imidazol-1-ylmethyl)piperidine
5-({2-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole