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N,N-diethyl-1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
(3R,5S)-N-[2-(2-chloro-6-fluorophenyl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
4-{4-[1-(3,4-dimethoxyphenyl)propan-2-yl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(2-methoxyphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(azocan-1-yl)-3-{5-[(cyclopentylamino)methyl]-2-methoxyphenoxy}propan-2-ol
N-{[1-(thiophene-3-sulfonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
[3-(1H-imidazol-1-yl)propyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3S,5R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
1-(oxane-4-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(1S,6R)-3-methyl-9-[3-(1H-pyrazol-1-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
1-{1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperazine
2-(dimethylamino)-2-(3-methylphenyl)-1-(thiomorpholin-4-yl)ethan-1-one
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[3-(2,5-dimethylfuran-3-yl)-1H-pyrazol-1-yl]acetamide
N-[2-(ethanesulfonyl)ethyl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propanamide
(5S)-5-[({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
methyl({[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(pyridin-4-ylmethyl)amine
N,3-dimethyl-4-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-3,4-dihydroquinazoline-7-carboxamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
N-{2-[2-(2,5-dioxoimidazolidin-4-yl)acetamido]-4-methylphenyl}benzamide
1-(1H-indazol-6-yl)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperazin-2-one
N-[(3,4-dimethoxyphenyl)methyl]-4-acetamido-N-(pyridin-2-ylmethyl)benzamide
7,7-dimethyl-2-[2-(4-methylpiperazin-1-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-bromo-5-(thiomorpholine-4-sulfonyl)benzoic acid
5-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
2-(furan-2-yl)-1-(3-propoxypropyl)-1H-imidazole
(1H-1,3-benzodiazol-2-ylmethyl)({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-{[(benzylsulfamoyl)amino]methyl}-N-ethyl-N-methylcyclohexan-1-amine
(4aS,8aR)-6-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
2-(3,4-dichlorophenyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}morpholine
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[4-(propan-2-yl)phenyl]urea
4,6-dimethyl-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
5-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylaniline
4-[2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-2-yl)ethyl]phenol
4-chloro-N,N-dimethyl-5-{1-[(2S)-oxolan-2-ylmethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]benzamide
2-({[3-hydroxy-2-oxo-1-(3-phenylpropyl)piperidin-3-yl]methyl}amino)-N-methylacetamide
3-{1-[6-amino-2-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-[1-(quinolin-2-ylmethyl)piperidin-3-yl]propanamide
1-cyclobutanecarbonyl-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
(4aS,8aR)-N-ethyl-1-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-4-(morpholin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
1-cyclopentyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-methanesulfonyl-N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-2-methylpyrimidin-4-amine