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3-(5-fluoropyridin-3-yl)-1-(oxan-4-yl)urea
9-[2-(3-methylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-(4-chloro-2-methylphenyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
3-methanesulfonamido-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(2,5-dioxoimidazolidin-4-yl)acetamide
9-(2-amino-2-methylpropanoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-{[1-(1H-imidazol-1-yl)propan-2-yl]amino}piperidin-1-yl)methyl]phenol
N-[(1R,3R)-3-aminocyclopentyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-phenoxyethan-1-one
1-[3-methoxy-5-(trifluoromethyl)phenyl]-3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)urea
2-{2-[(4-methyl-3-oxopiperazin-1-yl)methyl]-4-(pyrazin-2-yl)phenoxy}acetic acid
1-methyl-6-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indole
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
N-(2,6-dimethylphenyl)-3-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}benzamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(1H-pyrrol-1-yl)benzamide
4-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
2-cyclopropyl-9-(1-methyl-1H-pyrazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-{3-[4-(2-ethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
N-(2-methoxyethyl)-3-{[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]oxy}benzamide
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]urea
N-cyclopropyl-3-{1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]piperidin-3-yl}propanamide
1-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclobutan-1-amine
3-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(1,3-thiazol-2-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
6-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carbonitrile
4-{5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1,2,4-oxadiazol-3-yl}pyridine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amine
2-{[3-(furan-2-yl)-1-propyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-indazol-3-one
5-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,3-thiazol-2-amine
1-[1-(4-fluoro-3-methylbenzoyl)piperidin-4-yl]piperidin-3-ol
[1-(isoquinoline-5-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(pyridin-2-yl)propanamide
(2,1,3-benzoxadiazol-5-ylmethyl)({3-[1-(dimethylamino)ethyl]phenyl}methyl)methylamine
N-(2,3-dihydro-1H-inden-2-yl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-propylacetamide
1-amino-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)cyclopentane-1-carboxamide
1-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-N-methylpyrrolidine-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
5-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
4-({4-[(cyclopent-3-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-[5-({[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]carbamoyl}amino)-2-fluorophenyl]acetamide
5-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
4-[2-(4-chlorophenyl)morpholin-4-yl]-2-methoxypyridine-3-carbonitrile
3-chloro-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
N-[3-(aminomethyl)phenyl]-4-[2-(2-hydroxyethoxy)ethyl]piperazine-1-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-methoxy-2-methylpropan-1-one