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N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
2-methoxy-N-[3-({methyl[2-(2-methylpiperidin-1-yl)ethyl]carbamoyl}amino)phenyl]acetamide
N2-(2-methoxyethyl)-N4-[2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-{5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}morpholine
1-(1'-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
2-(2-methoxyphenyl)-5-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}piperidin-3-amine
1-(4-methoxyphenyl)-2,2-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)cyclopropane-1-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(4-methoxyphenyl)methyl]-3-(pyridin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-methyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
2-(2-chloro-6-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
{[(3R,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
7,7-dimethyl-2-{[2-(pyridin-3-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(2-oxo-2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-1,3-oxazolidin-2-one
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-[(5-propylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-({1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
methyl 3-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-4-methoxybenzoate
(3S,9aR)-8-benzyl-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{4-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]piperidin-1-yl}ethan-1-ol
4,6-dimethyl-2-oxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,2-dihydropyridine-3-carboxamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(dimethylamino)ethyl]acetamide
2-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
4-(3-methyl-1,2-oxazol-5-yl)-7-phenoxy-1,2,3,4-tetrahydroquinolin-2-one
2-methyl-6-[1-(thiolan-3-yl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
4-[2-(dimethylamino)ethoxy]-N-(4-phenylphenyl)piperidine-1-carboxamide
5-[1-(4-methoxyphenyl)cyclopropyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(1H-imidazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclohexyl-6-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,3-benzoxazole
N-[(2-chloro-4-fluorophenyl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-[4-({8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)phenyl]acetic acid
methyl 4-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]benzoate
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
2-methyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1,8-naphthyridine-3-carboxamide
2-(2-chlorophenyl)-3-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(4-chlorophenyl)-5-(3-methylthiophene-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{[(2H-1,3-benzodioxol-5-ylmethyl)(cyclopropyl)amino]methyl}pyridine-3-carboxylic acid
2-[2-(3-cyclobutyl-1,2,4-oxadiazol-5-yl)ethyl]-5-fluoro-1H-1,3-benzodiazole
4-methyl-2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
6-(4-methoxyphenyl)-N,7-dimethyl-N-(2-methylpropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
6-(3-chlorothiophene-2-carbonyl)-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
4-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]pyridine
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-phenyl-1,2-oxazole-3-carboxamide
1-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
(2S,4R)-4-amino-1-[5-(2-chlorophenyl)furan-2-carbonyl]-N-methylpyrrolidine-2-carboxamide
N-{3-[(6-ethylpyrimidin-4-yl)amino]propyl}-4-methylbenzene-1-sulfonamide
4-methyl-2-propyl-6-{4-[4-(pyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}pyrimidine
2-(propan-2-yl)-4-{1-[2-(pyridin-3-yloxy)propyl]-1H-imidazol-2-yl}pyrimidine