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2-[(4-phenylbutan-2-yl)amino]hexan-1-ol
[1-(1H-pyrazol-1-yl)propan-2-yl][2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]amine
N-({5-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N,N-diethyl-1-{5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}pyrrolidin-3-amine
6-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyridazin-3-amine
4-benzyl-3-[1-(1,4-dioxane-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methyl-1-phenylurea
4-(4-{[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyridazine
9-(2-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(3-chloro-1H-1,2,4-triazol-5-yl)propanamide
3-[3-(1H-pyrazol-3-yl)phenyl]pyrazine-2-carbonitrile
6-[(1,4-dioxan-2-ylmethyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-chloro-N-cyclopentyl-4-{[1-(1,3-dihydroxypropan-2-yl)piperidin-4-yl]oxy}benzamide
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-1H-indole
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
4-ethyl-1-methyl-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-6,7-dimethoxy-4-(oxolan-3-yl)-5H-indeno[1,2-b]pyridine-3-carbonitrile
1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-cyclopropylpiperidin-2-one
(3S,9aR)-8-(3-methoxybenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2-methoxyacetyl)-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}piperidine-3-carboxamide
6-{1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-cyclopropyl-6-(2-methylquinolin-5-yl)pyridazin-3-amine
N-ethyl-5-[(4-ethylpiperazin-1-yl)methyl]-N-propyl-1,2-oxazole-3-carboxamide
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-4-(thiophen-2-yl)butan-1-one
N,3,6-trimethyl-N-(1,2-oxazol-5-ylmethyl)-1-benzofuran-2-carboxamide
4-{3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzoyl}morpholine
1-[3-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]imidazolidin-2-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N1,5-bis(2-phenylethyl)piperidine-3,5-dicarboxamide
1-[4-(hydroxymethyl)pyridine-2-carbonyl]-4-methylpiperidine-4-carbonitrile
1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-{2-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
N-[2-(5-methylthiophen-2-yl)ethyl]-4-sulfamoylbenzamide
2-{1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperidin-4-yl}ethan-1-ol
4-{[1-methyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
[3-(cyclopropylmethyl)-1-(1,3-thiazol-2-yl)piperidin-3-yl]methanol
3-[3-(2-methylphenyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
3-(2-methylpropyl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1,2-oxazole-5-carboxamide
5-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1H-indole
8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-acetamido-1-(2-methoxyethyl)-2-(pyridin-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1H-1,3-benzodiazole-7-carboxamide
2-amino-N-[2-(1,3-benzothiazol-2-yl)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-ethyl-3-(1-ethyl-2-methyl-1H-indol-5-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]urea
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]propanamide
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
5-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-3-phenyl-1,2,4-oxadiazole