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N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-8-fluoroquinoline-2-carboxamide
methyl 3-{[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]carbamoyl}propanoate
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1,2,4-oxadiazol-3-yl)-1H-indole
1-[2-(cyclohex-1-en-1-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-[2-(pyridin-2-ylsulfanyl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(3-fluorophenyl)piperidine
1-[3-chloro-4-(propan-2-yloxy)phenyl]-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methylurea
N-(3-hydroxypropyl)-2-methyl-4-phenyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
N-[2-(2-ethoxyphenoxy)ethyl]-2-(4-methoxy-3-methylphenyl)-N-methylacetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[2-(methylsulfanyl)ethyl]amino}piperidin-1-yl)benzamide
4-{1-[(3-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-ethyl-5-methyl-1H-pyrazole
2-phenoxy-N-[1-({[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]acetamide
(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)-N-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]pyrrolidine-1-carboxamide
7-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-1,3-diazepane-2,4-dione
3-(azepane-1-carbonyl)-1-ethyl-N-[(2-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-2-yl)methanol
ethyl 1-({2-oxo-1-[2-(piperidin-1-yl)ethyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)piperidine-3-carboxylate
(3S,4S)-1-(1-aminocyclopentanecarbonyl)-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
5-(quinolin-8-yl)pyridine-2-carbonitrile
1-methyl-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-[3-cyclopropyl-5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
2-(2H-1,2,3-benzotriazol-2-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
N,N-dimethyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxamide
N-(5-{4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl}-1-(2-phenylethyl)-1H-1,3-benzodiazol-7-yl)-2-methoxyacetamide
3-{4-phenyl-5-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}propan-1-ol
4-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
1-benzyl-3-(2-methoxyethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(propan-2-yl)piperazine
5-[3-(5-methylfuran-2-yl)butyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-methyl-5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3,4-dihydropyrimidin-4-one
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-ethoxypropyl)acetamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-1-[(3-fluorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
(2S)-2-acetamido-N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(methylsulfanyl)butanamide
5-[1-(4-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
5-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-[2-(pyridin-3-ylformamido)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
4-(3-chloropyridin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[4-(1-ethyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-(5-fluoro-2-methylphenyl)propanamide
N-[2-(2-fluorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine