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1-cyclohexyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(pyridin-3-yl)propan-1-one
3-[(4-fluorophenyl)formamido]-N-methyl-N-[3-(oxolan-2-yl)propyl]propanamide
N-[2-(3-chlorophenyl)ethyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N,N-dimethyl-5-{[(5-methylfuran-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1'-(1,2,3,4-tetrahydroisoquinoline-6-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
5,6-dimethyl-2-(4-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-2-[4-(propan-2-yl)piperidin-1-yl]pyridine
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-2,2-dimethylpropan-1-one
1-[(3-chlorophenyl)methyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazine
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-3-methylbut-2-enamide
1-(3-chloro-2-ethoxyphenyl)-3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-methylurea
(2S,4S)-1-[2-(2,4-difluorophenyl)acetyl]-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
3-methyl-3-[(5-propyl-1H-pyrazol-3-yl)methyl]-1-[3-(sulfamoylmethyl)phenyl]urea
N-[2-methoxy-5-(methylcarbamoyl)phenyl]-3-(pyrimidin-4-yl)piperidine-1-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylurea
6-(benzyloxy)-1-cyclohexyl-4-(oxan-4-yl)-1,4-diazepan-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-hydroxyphenyl)acetamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N5-cyclopentyl-N3-ethyl-N3-(2-methylprop-2-en-1-yl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-ethoxy-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-hydroxyphenyl)ethan-1-one
(2S,4R)-1-(2-aminopyrimidin-4-yl)-N-(propan-2-yl)-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
4-[2-(3-hydroxyphenyl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(4-fluoro-3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(1,3-benzoxazol-2-yl)piperidin-4-amine
1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
5-(4-ethylpiperazin-1-yl)-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-amino-6-(methylamino)pyrimidin-4-yl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
6-{1-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-methoxy-N-({5-[2-methyl-2-(morpholin-4-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
4-(1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)thiomorpholine
(1S,5R)-3-[(2-methoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
14-(2-amino-1,3-thiazol-5-yl)-2,17-diazatetracyclo[9.8.0.03,8.013,18]nonadeca-1(19),3,5,7,11,13(18)-hexaen-16-one
5-(6-chloro-2H-chromen-3-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-[(3-fluorophenyl)methyl]piperazine
2-ethoxy-1-[6-hydroxy-4-(2-phenylethyl)-1,4-diazepan-1-yl]ethan-1-one
[(3,5-difluorophenyl)methyl](methyl){[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}amine
3-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propane-1,2-diol
3-methoxy-2-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
2-(3,4-dichlorophenyl)-4-(2-methylpyrimidin-4-yl)morpholine
2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}pyridine
ethyl 2-[4-(quinazolin-4-yl)piperazin-1-yl]-1,3-oxazole-4-carboxylate