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[1-(5-chloropyridin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
N,N-dimethyl-7-(4-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azetidin-3-yl}morpholine
1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-methyl-4-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
4-[(2-methoxyethyl)sulfamoyl]-N-(2-oxoazepan-3-yl)benzamide
(2R,3R)-3-[methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methylpropanamide
2-(4-hydroxybenzoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-2-yl)ethan-1-ol
1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
1-[6-(2,5-dimethoxyphenyl)pyridin-2-yl]piperazine
8-{[(4-methoxyphenyl)methyl]carbamoyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(5-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}thiophen-3-yl)methyl]dimethylamine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-methyl-3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-4,5,6,7-tetrahydro-1H-indazole
4-(1-butyl-1H-1,2,4-triazol-5-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
7-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-{4-[(5-methylfuran-2-yl)methyl]morpholin-3-yl}acetamide
N4-[(2,3-dimethyl-1H-indol-5-yl)methyl]pyrimidine-4,6-diamine
4-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}oxane-4-carbonitrile
3-{5-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-(naphthalene-1-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methylpyrimidin-2-amine
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
(3S,4R)-4-(3-fluorophenyl)-1-[3-(3-methoxyphenoxy)propyl]pyrrolidine-3-carboxylic acid
4-(3-{2-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-ylmethyl]phenoxy}propyl)morpholine
(2S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-acetamido-N,N-diethylpyrrolidine-2-carboxamide
N-methyl-2-(1,4-oxazepane-4-carbonyl)-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
2-(3-fluorophenyl)-5-(2-propoxyethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
methyl 3-[3-(cyclopentylcarbamoyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoate
5-[2-(trifluoromethyl)phenyl]pyrazin-2-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-hydroxy-1-(2-methyl-4-phenylpyridine-3-carbonyl)piperidine-4-carboxylic acid
N-(cyclopropylmethyl)-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)propanamide
5-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-(4-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
methyl (2S,4R)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-(2-phenylquinoline-4-amido)pyrrolidine-2-carboxylate
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(1,2-oxazolidin-2-yl)propanamide
(1R,3S)-1,3-dihydroxy-N-[(4-methylphenyl)methyl]-7-azaspiro[3.5]nonane-7-carboxamide
5-acetyl-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2,4-trimethyl-1H-pyrrole-3-carboxamide
1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
1-[2-(dimethylamino)ethyl]-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}pyrrolidin-2-one
2-({3-[(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)carbamoyl]phenyl}amino)acetic acid
(3R,5S)-5-[1-(2,3-dihydro-1H-inden-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyrrolidin-3-ol