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1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-4-yl)ethan-1-one
(3R)-N-(2,3-dimethylquinoxalin-6-yl)-3-hydroxypyrrolidine-1-carboxamide
2-{4-[1-(2-ethylbutyl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
N-(1H-indazol-5-yl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
(1R)-1-phenyl-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
3-methyl-N-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}but-2-enamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1-methyl-1H-imidazol-2-yl)piperidine
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-imidazol-2-yl)benzamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methylpyrimidin-2-amine
1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
4-(1-methanesulfonylpyrrolidine-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-(4-fluorophenoxy)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
2-(2,2-dimethyloxan-4-yl)-4-{3-[4-(2-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
3-(1-methyl-1H-imidazol-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(cyclopropylmethyl)-9-(2-methylpyridin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4-(1H-imidazol-2-yl)-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]piperidine
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
(3aR,7aS)-2-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-methoxy-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
3-(6-methoxynaphthalene-2-carbonyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
2-({[(1-ethylpyrrolidin-2-yl)methyl]amino}methyl)-8-fluoroquinolin-4-ol
2-methanesulfonyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[(3-ethyl-5-hydroxyadamantan-1-yl)formamido]-N-(1,3-thiazol-2-yl)propanamide
4-(2-methoxybutanoyl)-1-(2-methylphenyl)piperazin-2-one
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}(pyridin-3-ylmethyl)amine
4-(morpholin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-{4-[5-(pyrrolidine-1-carbonyl)furan-2-yl]phenyl}-1H-pyrazole
3-(1H-1,3-benzodiazol-1-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
ethyl 4-({[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
2-[1-(3-methylbutyl)-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl]ethan-1-ol
(1R,5R)-3-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(9H-purin-6-yl)-decahydro-1,6-naphthyridin-2-one
5-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)thiophene-2-carboxamide
(1S,4R)-2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2-azabicyclo[2.2.1]heptan-3-one
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}propanamide
2-{[methyl(propyl)amino]methyl}-N-(2-phenylethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)furan-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-methyl-5-phenyl-N-[2-(1,3-thiazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
7-(furan-2-ylmethyl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
3-(3-{octahydropyrrolo[1,2-a]piperazin-2-yl}propyl)-4,5,6,7-tetrahydro-2H-indazole
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(dimethylamino)acetyl]piperidin-4-yl}propanamide
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(pyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid