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N-benzyl-N-methyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-amine
1-(4-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}phenyl)-1H-1,2,3,4-tetrazole
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
4-ethyl-5-methyl-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-{2-[2-(methylcarbamoyl)-4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl]-2-oxoethyl}piperidine-4-carboxamide
9-[(4-fluoro-2-methylphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(methoxymethyl)piperidin-1-yl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[1-(4-ethyl-5-methylpyrimidin-2-yl)piperidin-4-yl]methanesulfonamide
2-phenyl-1-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}ethan-1-ol
2-[4-(2-ethyl-6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-1-yl]-2-oxo-N-(1,3-thiazol-2-yl)acetamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-{[1-(3-phenoxypropanoyl)pyrrolidin-3-yl]methyl}benzamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(4-methoxy-2-methylphenyl)-3-[1-(3-phenoxypropanoyl)piperidin-3-yl]propanamide
3-(furan-2-yl)-2-[2-(pyridin-3-yl)-1H-imidazol-1-yl]propanoic acid
N-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(quinolin-8-ylmethyl)amino]methyl}piperidin-2-one
3-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-{5-[3-(difluoromethoxy)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
6-[(diethylamino)methyl]-N-(2,4,6-trimethylpyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[2-(2,4-difluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
N-(2-methoxyethyl)-1-methyl-N-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}piperidin-4-amine
3-methyl-N-{2-[2-(thiophen-3-yl)-1H-imidazol-1-yl]ethyl}pyridin-2-amine
methyl 1-[2-hydroxy-3-(4-{[(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-(2H-1,3-benzodioxole-5-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-[(1S,5R)-6-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-{[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}spiro[azepane-4,2'-chromene]
8-{2-methylthieno[2,3-d]pyrimidin-4-yl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
4-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-2-(propan-2-yl)pyrimidine
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-methoxypyrazine
3-(1H-1,3-benzodiazol-2-yl)-1-[3-(3-methoxybenzoyl)piperidin-1-yl]propan-1-one
2-[5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1'-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S)-4-methyl-2-{[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]formamido}pentanamide
7-[(5-methylthiophen-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decane
N-{[3-methoxy-4-(pyridin-2-ylmethoxy)phenyl]methyl}-1-methyl-4-oxo-N-(oxolan-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
4-(1-benzofuran-5-ylmethyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
3-ethyl-5-(6-methoxy-3-methyl-1-benzofuran-2-yl)-1,2,4-oxadiazole
11-(morpholin-4-yl)-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,N-dimethyl-7-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
(3aR,6aR)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-{[2-chloro-5-(1H-pyrazol-1-yl)phenyl]formamido}acetamide
3-(3-chlorophenyl)-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one