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N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(morpholin-4-yl)pyridine-3-carboxamide
1-methanesulfonyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{3-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-oxopropyl}pyrrolidin-2-one
3-(hydroxymethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-propylpiperidine-1-carboxamide
N-benzyl-2-(dimethyl-1,3-thiazol-5-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]acetamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-(cyclohexylmethyl)pyrrolidine-2-carboxylate
1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidin-4-ol
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-phenylbenzoyl)pyrrolidin-3-yl]methanol
1-(3-chlorophenyl)-5-methyl-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
2-(2-methylfuran-3-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methylphenyl)acetamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]butanamide
3-{1-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
5-methoxy-1-methyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1H-indole-2-carboxamide
6-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-1,4-oxazepan-6-ol
4-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
(1R,2R)-1-[(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]-2,3-dihydro-1H-inden-2-ol
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(thiophene-3-carbonyl)pyrrolidine-2-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(3-hydroxypropyl)acetamide
2-[4-(azepan-1-ylmethyl)phenyl]-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-{2-hydroxy-3-[4-methoxy-2-({[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
2-{2-[1-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-ol
(1R,2R,4R)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetic acid
(1R,5S)-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-(6-aminopyrimidin-4-yl)-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-1,3-thiazole-4-carboxamide
8-benzoyl-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,2R,6S,7S)-4-(8-chloro-2-methylquinoline-4-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
2-(4-hydroxypiperidin-1-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
2-methoxy-5-sulfamoyl-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-4-phenoxybutan-1-one
N-cyclopropyl-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazine-2-carboxamide
1,9-dimethyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(4-methanesulfonylphenyl)-3-phenyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butanoic acid
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-ethyl-N-methyl-1,3,4-oxadiazol-2-amine
2-acetamido-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
N-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl]methanesulfonamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
1-cyclopentyl-4-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
3-(1-methyl-1H-pyrazol-4-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]propanamide
5-oxo-1-[2-(phenylamino)ethyl]pyrrolidine-3-carboxylic acid
3-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(propan-2-yl)-4-{4-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl}pyrrolidin-2-one
4-{[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]methyl}-1-(propan-2-yl)piperidine
(2S,4R)-4-acetamido-N,N-diethyl-1-[(3-fluoro-4-methoxyphenyl)methyl]pyrrolidine-2-carboxamide