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N-(adamantan-2-yl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
7-(5-chloropyridin-2-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(cyclooctylamino)methyl]-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
2-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-oxopropan-2-yl)-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
(4R)-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1,3-thiazolidine-4-carboxamide
2-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
3-[(3-{4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)methyl]phenol
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4-(dimethylamino)butanamide
N-(2-methoxyethyl)-5-methyl-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-cyclopropyl-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1,3,4-oxadiazol-2-amine
(3aS,7aR)-5-methyl-2-[2-(methylsulfanyl)benzoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-5-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(1-benzylpiperidin-4-yl)methyl]-2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methylacetamide
9-[(2-butyl-1H-imidazol-4-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]pyrimidin-2-amine
1-[4-(3-methylphenoxy)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
4-{[2-(azepan-1-yl)ethyl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-cyclopentyl-1-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
methyl 4-{[(2-{1-[1-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylpropanamide
methyl 4-{5-[(4-acetamidopiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoate
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(2-oxopyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-(1-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-yl}piperidine-3-carbonyl)piperazine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(2-methoxyphenyl)methyl]-N-methylacetamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
4-{[4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}phenol
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N-methylpyrimidin-2-amine
(1S,6R)-9-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
7-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2,3-dimethyl-1H-indole
1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(2S,4S)-4-amino-N-ethyl-1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)pyrrolidine-2-carboxamide
5-methoxy-1-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-indole-2-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-4-ol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
4-(4-chlorophenoxy)-N-[2-(dimethylamino)ethyl]piperidine-4-carboxamide
2-(1-benzyl-4-cyclohexylpiperazin-2-yl)ethan-1-ol
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
(1R,3S)-7-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
8-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3R,5S)-5-(methylcarbamoyl)-1-[2-(morpholin-4-yl)-2-oxoethyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-[2-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)phenoxy]ethan-1-ol
(3S,4S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
methyl 3-{[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}thiophene-2-carboxylate
N-{1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
3-methyl-8-[4-(1H-pyrazol-1-yl)butan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-ethylphenyl)-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)propanamide
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carboxamide
1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine