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2-(4H-1,2,4-triazol-4-ylmethyl)quinoline
2-{[1-(1-benzofuran-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-[2-(pyridin-3-yloxy)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(4,5-dimethyl-3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}thiophen-2-yl)-2-methylpropanamide
(3R,4R)-4-cyclobutyl-3-methyl-1-(pyridin-4-yl)piperidin-4-ol
2-[(2,6-dichlorophenyl)methyl]-5-(4-ethylpiperazine-1-carbonyl)pyrimidin-4-ol
3-[2-(piperidin-2-yl)ethyl]-5-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]phenol
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
4-oxo-1-(2-phenylethyl)-5-[(thiolan-3-yl)carbamoyl]-1,4-dihydropyridine-3-carboxylic acid
4-{1-[1-(2,2-diphenylethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
1-(2-methoxyethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrrolidine-3-carboxamide
2-(4-chlorophenyl)-5-[1-(3-methoxypropyl)-1H-imidazol-2-yl]pyrimidine
(1S,5R)-3-(2,1,3-benzothiadiazol-5-ylmethyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-cyclopentyl-4-[(3,5-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(2S)-2-amino-3-hydroxy-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
2-(2-methoxyphenoxy)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
N-methyl-3-(5-methylfuran-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
6-(azocan-1-yl)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
2-methoxy-4-(quinolin-8-yl)pyridine-3-carbonitrile
N-[2-(1,3-benzothiazol-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
[(4-methanesulfonylphenyl)methyl](methyl){[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-[(4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-N,N-dimethylaniline
8-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
3-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-1-[(5-methyl-1,2-oxazol-3-yl)methyl]urea
1-(4-chlorophenyl)-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
4-[(2-ethoxyphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
(1R,9aR)-1-{[3-(pyridin-3-yl)-1H-pyrazol-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
2-[3-(pyrrolidin-1-yl)pyrazin-2-yl]benzonitrile
3,5-dimethyl-2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-1H-indole
1-(2-{[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}-4-methylpyrimidin-5-yl)ethan-1-one
N-(3,4-dimethylphenyl)-2-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}amino)acetamide
N'-(1,3,4-thiadiazol-2-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]butanediamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
1-benzyl-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[1-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)piperidin-3-yl]benzoic acid
2-amino-6-(4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
4-phenyl-N-[4-(propylcarbamoyl)phenyl]piperidine-1-carboxamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(thian-4-yl)piperazine
2-{[5-(2-methoxyphenyl)-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
7-chloro-N-(dimethyl-1H-1,2,4-triazol-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
2-methyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]-1-(propan-2-yl)piperazine
2-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxo-N-propylacetamide
5-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
1-(2,3-dihydro-1H-inden-2-yl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-amine
N,N-dimethyl-2-(6-{[2-(morpholin-4-yl)ethyl]amino}pyridin-3-yl)benzamide