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3-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2,2-dimethylpropan-1-ol
3-[2-(adamantan-1-yl)acetamido]-N-(2-fluorophenyl)propanamide
7-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
(3S,4S)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-[(2-methoxyethyl)(methyl)amino]pyrrolidin-3-ol
6-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
2-(2-fluorophenoxy)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}ethane-1-sulfonamide
[(4-methanesulfonylphenyl)methyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
2-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-4-carbonitrile
2-amino-N,4-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
1-{3-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-N-(3-chloro-4-methoxyphenyl)propanamide
1-{6-hydroxy-4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,4-diazepan-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
3-butyl-5-(3-chlorothiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]pyridine-3-carbonitrile
4-({5-[(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
1-[6-hydroxy-4-(oxan-4-yl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
3-(3-fluorophenyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)-1H-pyrazole-4-carboxamide
N-[3-(dimethylamino)propyl]-N-methyl-1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-3-amine
N-(1-benzothiophen-2-ylmethyl)-6-{[benzyl(butyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(3-chloro-5-fluorobenzoyl)-1-(3,5-dimethylphenyl)piperazin-2-one
1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-{5-[(2-ethylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-[2-(dimethylamino)ethyl]-5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
9-[3-(3-fluorophenyl)propanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
5-(morpholin-4-yl)-2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
N-[3-(1H-imidazol-5-yl)phenyl]-4-methanesulfonylpiperazine-1-carboxamide
7-cyclopentyl-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclopentyl-2-methoxy-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxypropan-1-one
2-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
9-methoxy-N-[(4-methoxyphenyl)methyl]-3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)acetamide
(4aR,8aR)-4a-hydroxy-7-{imidazo[1,2-a]pyridine-6-carbonyl}-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-ethyl-2-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-1-yl]pyrimidin-4-amine
1-(4-methoxyphenyl)-3-[1-methyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]propan-1-one
4-[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-6-(propan-2-yl)pyrimidine
5-ethyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-[1-(4-cyanopyridin-2-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
4-cyclobutyl-N-(1-ethylpiperidin-3-yl)-6-methylpyrimidin-2-amine
N-[2-(methylsulfanyl)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
(2S,4S)-4-amino-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-(morpholin-3-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
(3R,5S)-5-(morpholin-4-ylmethyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-(2-phenylethyl)piperidine-3-carboxamide
1-(carbamoylmethyl)-N-{[5-chloro-2-(propan-2-yloxy)phenyl]methyl}piperidine-3-carboxamide