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7-[5-(oxolan-2-yl)thiophene-2-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
8-chloro-2-({[3-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)quinolin-4-ol
(3R)-1-({1-[1-(furan-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
4-amino-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-2-one
(3aR,6aR)-2-[4-(1H-imidazol-1-yl)butanoyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1H-imidazol-2-ylmethyl)-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
3-(2-methoxybenzoyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-oxopiperidin-3-yl)-1,3-oxazole-4-carboxamide
7-amino-4-[4-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-[(2-fluorophenyl)methyl]-N-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-3-amine
2,3,4-trimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
4-(1H-imidazol-1-yl)-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]benzamide
1-(2-{[(1-benzyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-{1-cyclopentyl-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-5,6-dimethylpyrimidin-2-amine
N-(3-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-2-methylphenyl)furan-2-carboxamide
1-(4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)propan-1-one
N-[2-(4-chlorophenyl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-(oxolan-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
7-methoxy-3-(4-methylpiperazine-1-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-(furan-2-ylmethyl)-4-[1-(oxan-4-yl)piperidine-4-carbonyl]piperazine
9-[(3-hydroxyphenyl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(oxan-4-yl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
2-(4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)-1,3-benzoxazole
4-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-(2-phenylethyl)-4-{spiro[2.5]octan-1-ylmethyl}piperazine
propan-2-yl 4-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carboxylate
N-[2-(morpholin-4-yl)ethyl]-4-(4-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}piperidin-1-yl)benzamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
6-(4-oxo-4H-chromene-2-carbonyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
methyl 6-{[4-(2-methylpropyl)phenyl]methyl}-2-(morpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(2-methoxy-4-propylphenoxy)-1-azabicyclo[3.2.1]octane
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(dimethylamino)ethyl]-3-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}propanamide
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
4-(7-chloroquinolin-4-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenol
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazole
1-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2-methylphenol
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
10-methoxy-5-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-benzyl-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-(azepan-1-yl)-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide