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N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(morpholine-4-sulfonyl)benzamide
N-cyclohexyl-N-[(4-fluorophenyl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]-2-ethylpyrimidine
N-(oxolan-3-yl)-4-{[2-(1H-pyrrol-1-yl)ethyl]sulfamoyl}benzamide
methyl (2S)-1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]pyrrolidine-2-carboxylate
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyridin-4-yl)propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-amino-4-[2-(benzylamino)pyrimidin-5-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
benzyl(benzylsulfamoyl)[2-(dimethylamino)ethyl]amine
3-(2-aminoethyl)-4-(2H-1,3-benzodioxol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopentyl-N-ethyl-3-(3-hydroxy-3-methylbutyl)benzamide
7-chloro-2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-4-methylquinoline
N-[1-(hydroxymethyl)cyclopentyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-butyl-4-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-6-methylpyrimidin-2-amine
(1-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
2-amino-6-(3,5-difluorophenyl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-4-(pyrazin-2-yl)piperazine-1-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(3-fluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2H-1,3-benzodioxol-5-yl)-N-tert-butyl-3-phenylpropanamide
2-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[2-(5-methylthiophen-2-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(thiophen-2-yl)acetamide
(2S)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-oxopyrrolidine-2-carboxamide
3-methoxy-5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridine
2-(2,4-dichlorophenoxy)-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]ethan-1-one
(2S,4S)-4-benzamido-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
(4aS,8aR)-6-(3-methylfuran-2-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-({[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)-4H-chromen-4-one
3-methoxy-2-[(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
6-methoxy-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrimidin-4-amine
4-(piperidin-3-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-{3-cyclopropyl-5-[2-(1H-imidazol-4-yl)-1-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
N4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]pyrimidine-4,6-diamine
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-ol
(3S,4S)-1-[(2-cyanophenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
3-(3-fluorophenyl)-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazin-2-one
1-{4-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
(3S,4S)-1-{2-[benzyl(ethyl)carbamoyl]ethyl}-4-cyclopropylpyrrolidine-3-carboxylic acid
(2S)-1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxy-3-phenylpropan-1-one
6-[({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)methyl]-1,4-oxazepan-6-ol
1-[3-(furan-2-yl)propanoyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-(2-chloroprop-2-en-1-yl)-3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
8-methoxy-2-methyl-5-[5-(morpholine-4-carbonyl)furan-2-yl]quinoline
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1-propylpiperidin-4-yl)piperidine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[phenyl(pyridin-4-yl)methyl]acetamide
2-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidin-2-yl}pyridine
N-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-amine