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N-[4-(3-methylphenyl)phenyl]-1-(4,4,4-trifluorobutanoyl)piperidine-4-carboxamide
1-{3-carboxy-5H,6H,7H-cyclopenta[b]pyridin-2-yl}-4-phenoxypiperidine-4-carboxylic acid
2-{1-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-4-methyl-1,3-thiazole
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-cyclopentyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N4,N4-dimethyl-N2-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
ethyl 4-{1-[(6-chloro-2H-chromen-3-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2-dihydrophthalazin-1-one
methyl 1-{[4-(1-benzyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
4-{[1-(1H-pyrazole-4-carbonyl)piperidin-2-yl]methyl}morpholine
4-(2-methylpropyl)-1-(2,3,4-trifluorobenzoyl)-1,4-diazepan-5-one
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)pyridine-3-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
4-cyclopentyl-3-oxo-N-[4-(oxolan-2-ylmethoxy)phenyl]piperazine-1-carboxamide
4-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-methylpyrrolidin-2-one
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(oxane-4-carbonyl)piperidin-3-ol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-4-sulfamoylbenzamide
1-[1-(3-methoxypropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-[ethyl(methyl)amino]-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-[2-(dimethylamino)ethyl]-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-2-butyl-5-chloro-1H-imidazole
(5-{2-[(dimethylamino)methyl]phenoxy}-2,3-dihydro-1-benzofuran-2-yl)methanamine
(3S,4S)-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
(2R,6R)-11-methoxy-4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-methyl-5-{1-[1-(6-methylpyridin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}quinoline
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)thiophene-3-sulfonamide
1-ethyl-3-({4-[2-(methylsulfanyl)propyl]-1H-1,2,3-triazol-1-yl}methyl)-1H-indazole
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]pyridine-4-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(6-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
(4aR,7aS)-1-methyl-4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopentyl-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N'-(3,5-dimethylphenyl)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]propanediamide
2-({[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenol
8-[4-(1H-indol-3-yl)butan-2-yl]-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3,4-dimethoxyphenyl)methyl]-1-ethyl-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-7-yl}-1H-1,2,4-triazole
(1S,5R)-6-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]pyrimidine-5-carboxamide
1-(4-ethoxy-3-methylphenyl)-4-[4-(propan-2-yl)piperazin-1-yl]butane-1,4-dione
2-ethoxy-1-{6-methyl-5-[5-(1-methyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
5-cyclobutanecarbonyl-1'-(pyrrolidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(5S,9aS,9bS)-5-[3-(methylsulfanyl)phenyl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
{4-[(4-methoxyphenyl)methyl]-1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}methanol
5-(1-ethyl-6-oxopiperidine-3-carbonyl)-N,N-dimethyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
5-cyclopropyl-N-(2-hydroxyethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-[4-(benzyloxy)piperidine-1-carbonyl]pyridine-2-carbonitrile
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(2-oxopyrrolidin-1-yl)acetamide