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1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{4-[({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)methyl]phenyl}cyclopropanecarboxamide
2-(2-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1-(4-benzylpiperidin-1-yl)propan-1-one
N-[(7-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
[(3R,4R)-1-(1H-imidazol-2-ylmethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
6-ethyl-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[5-methoxy-2-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
{imidazo[1,2-a]pyridin-3-ylmethyl}({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-3-(1H-pyrazol-4-yl)propanamide
(3R,4R)-3,4-dimethyl-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-ol
2-(2,2-dimethylpropanamido)-5-methyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]thiophene-3-carboxamide
9-[(3,5-dimethylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(4-phenoxyphenyl)methyl]oxane-4-carboxamide
1-(furan-2-yl)-2-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}ethane-1,2-dione
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(4-methoxybenzoyl)piperazine
5-methyl-3-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-2-yl]-1,2-oxazole
4-{4-[(2,3-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-(2-fluorophenyl)piperidin-4-ol
(3S,4R)-1-(2,3-difluoro-4-methylbenzoyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
8-(3-hydroxypyridine-2-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methoxyphenyl)methyl]piperidine
2-methyl-4-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenol
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-(2-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-oxoethyl)imidazolidine-2,4-dione
2-{[1-(2,6-dimethylphenoxy)propan-2-yl]amino}-N-(pyrazin-2-yl)acetamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl]methanol
N-cyclohexyl-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(2S)-2-amino-3-methoxy-N-[2-(3-oxopiperazine-1-carbonyl)phenyl]propanamide
1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
2-{3-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]phenoxy}acetamide
5-ethyl-5-{1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(3-hydroxy-3-methylbutyl)-N-[1-(hydroxymethyl)cycloheptyl]benzamide
N-[3-methoxy-4-(3-methylbutanamido)phenyl]-1H-indole-5-carboxamide
1-[(4aR,8aS)-6-(3-phenylpropyl)-decahydro-1,6-naphthyridin-1-yl]ethan-1-one
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1-benzothiophene-5-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}[(2-phenoxypyridin-3-yl)methyl]amine
(3R,9aR)-3-(propan-2-yl)-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
6-(cyclopropylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2,5-dimethylphenyl)methyl]propanamide
N-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(4aR,6R,8aS)-2-benzyl-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-(3-ethoxyphenyl)-4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carboxamide
3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-4-fluorobenzene-1-sulfonamide
5-chloro-N-methyl-2-oxo-N-(quinolin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
3-(2-chlorophenyl)-3-phenyl-N-[2-(piperazin-1-yl)ethyl]propanamide