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4-({4-[2-(3-methoxypiperidine-1-carbonyl)-4-methylphenoxy]piperidin-1-yl}methyl)pyridine
1,9-dimethyl-N-[4-(methylsulfanyl)phenyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(4aR,7aS)-1-methanesulfonyl-4-(5-methylpyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
(1R,5S,8S)-3-[(2,3,4-trimethoxyphenyl)methyl]-3-azabicyclo[3.2.1]octan-8-ol
1-{6-[3-(1H-pyrazol-3-yl)phenyl]pyridin-3-yl}ethan-1-one
2-[1-cyclopentyl-4-(6-methylpyridazin-3-yl)piperazin-2-yl]ethan-1-ol
3-benzyl-4-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperazin-2-one
1-[(3-{[1-(4-methylbenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N3-[2-(3-propoxyphenyl)ethyl]piperidine-1,3-dicarboxamide
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-imidazole
2-(cyclohex-1-en-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-methyl-6-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
5-cyclobutyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
{[5-(1-cyclopentanecarbonylpiperidin-4-yl)-4-ethyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
(3aR,6aR)-2-cyclopentyl-5-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3-{2-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-[(3-chlorophenyl)methyl]-4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazine
2-(propylsulfanyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-(1H-pyrazol-5-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
4-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-2-ethyl-1-(propan-2-yl)piperazine
N-[(3,4-difluorophenyl)methyl]-3-[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
3-(2-phenylethyl)-5-[(phenylsulfanyl)methyl]-1H-1,2,4-triazole
5-(4-methoxy-2-methylphenyl)pyridin-2-amine
2-[methyl({[4-methyl-5-(1-methylpiperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]ethan-1-ol
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1R,6S)-9-methyl-3-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonane
4-methyl-N-propyl-N-(pyridin-4-ylmethyl)-1H-imidazole-5-carboxamide
8-[(3,5-dichloropyridin-4-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-(azocan-1-yl)-N-[3-(pyridin-3-yl)propyl]propanamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
3-phenoxy-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
(4aS,7aR)-1-(3-chloro-4-methoxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methyl-1,2-oxazole-5-carboxamide
N-[(4-methoxyphenyl)methyl]-2-(2-oxopiperidin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
2-({4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-1,2,3,4-tetrahydroisoquinoline
N6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-9H-purine-2,6-diamine
N-[2-(4-{[(1H-indol-3-ylmethyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]methanesulfonamide
3-fluoro-N-({7-[4-(pyrrolidin-1-yl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3,6-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]amine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(3,5-dimethyl-1H-pyrrol-2-yl)-3-(methoxymethyl)-1,2,4-oxadiazole
8-{[2-(furan-2-yl)phenyl]methyl}-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-ethyl-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)benzamide
2-[2-(2-fluorophenyl)ethyl]-4-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide