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dimethyl[2-(2-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
methyl 4-(5-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(3R,4R)-3-{ethyl[(2E)-3-(furan-2-yl)prop-2-en-1-yl]amino}-4-hydroxy-1λ6-thiolane-1,1-dione
(4aS,8aR)-6-(6-methoxypyrimidin-4-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[2-(cyclohexylformamido)ethyl]-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-({2-[3-(dimethylamino)propoxy]-3-methoxyphenyl}methyl)azepan-4-ol
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-4-ol
1-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
(1H-indol-2-ylmethyl)(methyl)[3-(pyrrolidin-1-yl)propyl]amine
N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyrazin-2-ylmethyl)pyridin-2-amine
5-(1-cyclohexanecarbonylpyrrolidine-2-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-oxo-4-phenylbutanamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]acetamide
3-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4-(1H-pyrazol-3-yl)benzamide
(1S,5R)-3-(3-chloro-4-hydroxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(2-fluorophenyl)methyl]-6-(5-oxopyrrolidine-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(2R,6R)-4-(5-hydroxypyrazine-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2R,3R)-1'-[2-(hydroxymethyl)pyridin-4-yl]-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(3S)-3-ethyl-4-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]morpholine
1-(4-chlorophenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]cyclobutane-1-carboxamide
3-[(cyclohex-3-en-1-ylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(phenylsulfamoyl)benzamide
N-[(2-fluorophenyl)methyl]-5-[1-(3-methoxypropanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[5-(methoxymethyl)furan-2-carbonyl]-decahydro-1,6-naphthyridin-2-one
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(carbamoylmethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1-phenylpiperazin-2-one
3-[(2R)-2-amino-2-phenylacetamido]-N-(2-methylphenyl)propanamide
(4-{[(5-ethylpyrimidin-2-yl)(methyl)amino]methyl}oxan-4-yl)methanol
6-methyl-2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]pyridine-3-carboxylic acid
3-benzyl-4-(4-hydroxybenzoyl)piperazin-2-one
N-(2-hydroxyethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
2-(cyclopropylmethyl)-9-(3-hydroxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-amino-7-(5-hydroxypyrazine-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-methyl-2-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,8-diazaspiro[4.5]decan-3-one
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-(1,4-dioxan-2-ylmethyl)-2,4-dimethoxybenzamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(1H-indazol-1-yl)propyl]acetamide
2-fluoro-N-{1-[({[1-(piperidin-1-yl)cyclohexyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}benzamide
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-2-methyl-1,4-diazepan-5-one
N-(3,5-dimethoxyphenyl)-3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanamide
4-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
8-benzyl-3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,4S)-4-hydroxy-1-phenylmethanesulfonylpiperidine-2-carboxylic acid
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(methylsulfanyl)propan-1-one