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N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2,4-dichlorophenoxy)-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]acetamide
(4-{[1-(4-aminopyrimidin-2-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
(3R,5S)-N-[(3,4-difluorophenyl)methyl]-1-(pyridin-3-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
2-{[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}-N-cyclopropylacetamide
1-[2-methoxy-5-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-(oxolan-3-yl)-5-[5-(propan-2-yl)-1,3-oxazol-4-yl]-1,2,4-oxadiazole
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
N-[2-(4-fluorophenyl)ethyl]-5-{1-[(4-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-1-benzofuran-2-carboxamide
1-(1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-3-methylbutan-1-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(1-methylcyclopropanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-methyl-2-(methylamino)propanamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
6-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)acetamide
N-[3-(2-methoxyethoxy)phenyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
2,4-dimethyl-3-oxo-N-{4-[2-(pyridin-2-yl)ethoxy]phenyl}piperazine-1-carboxamide
N-methyl-6-{[(5-methylpyrazin-2-yl)methyl]amino}-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepane
N-tert-butyl-2-[5-(dimethylamino)-1-ethyl-1H-1,2,4-triazol-3-yl]benzene-1-sulfonamide
3-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[3-(1H-indol-1-yl)propyl]pyrimidin-4-amine
N'-[2-(propan-2-yl)phenyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]butanediamide
7-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
methyl 1-({6-[methyl(2-phenylethyl)carbamoyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-2-carboxylate
(4aS,8aR)-6-[3-(furan-2-yl)propanoyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
4-(2,3-dimethylquinoxaline-6-carbonyl)-1-methylpiperazin-2-one
N,N-dimethyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]({[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl})methylamine
N-(3-methoxypropyl)-1-methyl-N-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-amine
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-cyclopropyl-3-(oxan-4-yl)-1H-1,2,4-triazole
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(oxolane-2-carbonyl)piperazine
N-(2-chlorophenyl)-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
(4aS,8aR)-1-(3-methylbutyl)-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
(5-{1-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
2-(methoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(pyridin-2-yl)-7-(4,4,4-trifluorobutanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3R,4S)-4-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-1-yl}oxolan-3-ol
5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-2,1,3-benzoxadiazole
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
1-{1-[(3-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl}-4-methylpiperazine
9-methoxy-7-(5-methylthiophen-2-yl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-ethoxypropan-1-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(3-hydroxyadamantan-1-yl)acetamide