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N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2,3,6-trimethylphenoxy)acetamide
1-(2-methoxyethyl)-3-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-1-(pyridin-4-ylmethyl)urea
N-(1-benzylpiperidin-4-yl)-5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-(2-hydroxy-2-phenylethyl)-N-(pyridin-4-ylmethyl)acetamide
3-[(4aR,7aS)-4-(cyclopentylcarbamoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
6-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide
(4-{[2-(furan-2-yl)phenyl]methyl}morpholin-2-yl)methanamine
7-[(3,4-difluorophenyl)methyl]-2-(1H-imidazol-2-ylmethyl)-2,7-diazaspiro[4.5]decane
ethyl 1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
5-methoxy-2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1H-indole
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(4-{2-methoxy-5-[2-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
5-(2-chlorophenyl)-N-(2-methoxyethyl)-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]furan-3-carboxamide
3-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3-(1-methylcyclopropyl)propan-1-one
(4aS,8aR)-1-(2-methylpropyl)-6-[(6-methylpyridin-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-3,6-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
5-{2-[2-(9H-fluoren-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2-dimethyl-1H-1,3-benzodiazole-5-carboxamide
(4aR,7aS)-1-butyl-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3,4-dimethylpiperidin-4-ol
2-(4-fluorophenyl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-hydroxyethan-1-one
(2-{3-cyclopropyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}ethyl)urea
[2-(cyclohex-1-en-1-yl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
2-ethyl-4-{[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}pyrimidine
(2S,4R)-4-amino-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-methylpyrrolidine-2-carboxamide
{3-[5-(4-chloro-2-fluorophenyl)-4-phenyl-1H-imidazol-1-yl]propyl}(methyl)amine
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
8-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-fluorobenzene-1-sulfonamide
5-methoxy-1-methyl-2-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-indole
(1S,5R)-3-(1H-1,2,3-benzotriazole-5-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
4-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[4-(2-fluorophenoxy)phenyl]-1-(thiophen-2-ylmethyl)piperidine-4-carboxamide
5-ethyl-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(methoxymethyl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}cyclobutane-1-carboxamide
4-(naphthalen-1-yl)-3-(oxan-4-yl)-4H-1,2,4-triazole
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
1-cyclohexyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
1-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
(2R)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-acetamidopropanamide
3-[(2-hydroxyethyl)[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]amino]-1λ6-thiolane-1,1-dione
2-[(4-chlorophenyl)sulfanyl]-1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
methyl 5-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}pentanoate
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-4-(trifluoromethyl)pyrimidin-2-amine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]oxolane-2-carboxamide
4-(1-hydroxy-2-phenylethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide