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N1-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]pentane-1,5-diamine
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-(hydroxymethyl)-N-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]piperidine-1-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-butyl-1-cyclohexyl-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[1-(4-methanesulfonylphenyl)propyl]-1-methyl-1H-indole-6-carboxamide
1-cyclohexanecarbonyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-({2-[(2-methylpyrrolidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-2-phenyl-1,3-oxazole
3-[(2-methoxyethyl)(methyl)sulfamoyl]-N-methyl-N-(pyrazin-2-ylmethyl)benzamide
N-(furan-2-ylmethyl)-2-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
5-ethyl-N-[1-(4-methanesulfonylphenyl)propyl]-1,3,4-oxadiazol-2-amine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
(2S)-3-methyl-2-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)butan-1-ol
9-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-3-methoxy-1-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]piperidin-4-amine
methyl({[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
1-[4-(benzenesulfonyl)piperazin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazole
5-methyl-1'-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-methoxy-3-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-indole-2-carboxamide
(2S)-1-acetyl-N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
2-({2-[2-(propan-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}methyl)-1,3-benzothiazole
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(3-methoxyphenyl)propanoyl]-decahydro-1,6-naphthyridin-2-one
5-methyl-1-(4-methylphenyl)-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidin-2-one
5-butyl-N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]pyridine-2-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl](ethyl)(pyridin-3-ylmethyl)amine
4-[(2-fluoro-5-methoxyphenyl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-{1-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
3-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)propanamide
2-({[(3R,4R)-1-(4-chloro-2-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
1-[(3-fluorophenyl)methyl]-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
2-methoxyethyl 4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
5,6-dimethyl-2-[2-oxo-2-(3-oxo-4-phenylpiperazin-1-yl)ethyl]-2,3-dihydropyridazin-3-one
5-methyl-N-{3-[(pyridin-3-yl)amino]propyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-N-(quinolin-5-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{2-[methyl(phenyl)amino]propyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-ethoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
7-(3-chlorophenyl)-4-cyclobutanecarbonyl-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-(1H-indol-2-ylmethyl)-6-(methoxymethyl)pyrimidin-4-amine
2-(2-aminoethyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}quinazolin-4-amine
(3aR,6aS)-5-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid