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N-[(3R,4S)-1-(3-cyano-6-methylpyridin-2-yl)-4-cyclopropylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
3-(3-hydroxy-3-methylbutyl)-N-{[(1r,4r)-4-(hydroxymethyl)cyclohexyl]methyl}benzamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N,6-dimethylpyrimidin-4-amine
2-[3-benzyl-1-(4-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclobutylacetamide
(1S,5R)-6-(2-methoxyethyl)-3-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,3-dihydroxypropyl)-N-methyl-4-propylpyrimidine-5-carboxamide
3-[4-(2-ethylphenyl)piperazine-1-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane
N-[(2S,4R,6S)-2-(2-phenylethyl)-6-{pyrazolo[1,5-a]pyrimidin-3-yl}oxan-4-yl]acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamide
4-(4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)morpholine
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)propanamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-(piperazin-1-ylmethyl)piperidin-2-one
2-fluoro-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-N-(4-methoxyphenyl)piperidine-1-carboxamide
ethyl 4-{[1-(4-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)piperidin-4-yl]amino}piperidine-1-carboxylate
2-{3,5-dimethyl-4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-1H-pyrazol-1-yl}ethan-1-ol
2-(dimethylamino)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-(3-methylphenyl)acetamide
N-cyclopropyl-5-methyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
3-{5-[2-(diethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-1-[(1R,2S)-2-(methoxymethyl)cyclopentyl]urea
4-benzyl-3-ethyl-1-[2-(piperazin-1-yl)acetyl]-1,4-diazepan-5-one
N-cyclopropyl-3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
5-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
2-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}acetic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-chloro-5-acetamido-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-(2-hydroxyethyl)-8-(2-methyl-2-phenylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aR,5S,6S,7aS)-2-{[3-(5-methylfuran-2-yl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-(4-methyl-5-{[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]sulfonyl}-1,3-thiazol-2-yl)acetamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
11-[4-(diethylamino)-2-ethoxyphenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
5-(2-chlorophenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]furan-2-carboxamide
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-(2,2,2-trifluoroethyl)propanamide
4-[5-(1-methylpyrrolidin-2-yl)thiophene-2-carbonyl]morpholine
6-tert-butyl-N,1-dimethyl-N-(oxan-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-6-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-(2H-1,3-benzodioxol-5-yl)-N-ethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
8-(2-phenylquinolin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[2-(pyrrolidin-3-yl)benzoyl]piperidine
ethyl 4-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)piperidine-1-carboxylate
ethyl 4-{2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamido}piperidine-1-carboxylate
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
2-methoxy-1-{1'-[(1r,4r)-4-methylcyclohexanecarbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
4-(3-acetylphenyl)-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
3-ethyl-N-[(2R)-oxolan-2-ylmethyl]-1H-indole-2-carboxamide
1-cyclohexyl-N3-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N3,N5-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide