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5-(2-fluoro-6-methoxyphenoxymethyl)-3-(phenoxymethyl)-1,2,4-oxadiazole
4-(2,6-difluorophenyl)-5-[(3-ethenylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-(2-fluorophenyl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-[(methylsulfanyl)methyl]pyridine
N-[1-({[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
5-{2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-ethoxypyridine-3-carboxamide
4-(hydroxymethyl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidin-4-ol
1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]-2,3-dihydro-1H-indole
6-(6-methoxypyridin-3-yl)-N,N-dimethylpyrazin-2-amine
4-{[3-(4-phenylbenzoyl)piperidin-1-yl]methyl}pyridine
[(3R,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
5-(3,4-dichlorophenyl)pyrimidine
(3S,4R)-N,N-dimethyl-1-[4-(2-methylpropyl)benzoyl]-4-propylpyrrolidin-3-amine
2-[2-(butan-2-yl)phenoxy]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]acetamide
3-[2-(5-propylfuran-2-yl)-1H-imidazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(5-{[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{4-[(1-methylpiperidin-3-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
2-(2-methoxyethyl)-9-(4-propylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-phenyl-2-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]propanoic acid
2-amino-6-(4-fluorophenyl)-5-methyl-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
5-(4-fluorophenyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
[(3-cyclopropyl-1H-pyrazol-5-yl)methyl][1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]methylamine
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
(3aR,7aS)-2-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
2-(1H-1,3-benzodiazol-1-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
5-ethyl-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}pyrimidin-2-amine
2-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-2-yl)acetic acid
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(thian-4-yl)piperazine
3-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl](methyl)amino}-N-methylpropanamide
2-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-1-[(3R)-pyrrolidin-3-yl]urea
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-cyclopropanecarbonyl-1'-[(3-ethoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-[2-(2-aminoethyl)quinazolin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
3-{6-amino-5-cyano-4-[2-(ethylamino)pyrimidin-5-yl]pyridin-2-yl}benzoic acid
1-(2-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4-methyl-1H-1,2,3-triazole
N-methyl-3-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]sulfamoyl}-N-(2-methylpropyl)benzamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-hydroxyethan-1-one
2-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,2-oxazinane
(3S,4R)-1-(2-carbamoylethyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(azepan-1-yl)-2-phenylethyl]propanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylcyclopropanesulfonamide
2-(2-phenylethyl)-9-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one