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9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1'-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-methyl-2,7-diazaspiro[4.5]decane
(3S)-N-tert-butyl-2-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-2-yl]pyridine
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
2-[4-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)morpholin-2-yl]ethan-1-ol
1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
3-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
N1,N1-dimethyl-N4-[(3-phenylphenyl)methyl]piperidine-1,4-dicarboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(1-cycloheptylpiperidin-3-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-phenyl-7-[2-(piperidin-1-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2,8-dimethyl-4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}quinoline
N-cyclopropyl-2-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyridine-4-carboxamide
2-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
ethyl 2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
4-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}piperazin-2-one
N-(propan-2-yl)-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methylpentan-1-one
5-[(1-benzylpiperidin-4-yl)amino]-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-methyl-8-[2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-4-(pyridine-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[(2R,3R)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pyrazine-2-carbonitrile
(2-methoxyethyl)[(4-methylphenyl)methyl](1,3-thiazol-2-ylmethyl)amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
3-methyl-4-[2-(3-methylphenyl)pyrimidin-5-yl]-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-[(3-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methoxy]-2-methyl-1,3-benzothiazole
3-{5-[2-(dimethylamino)-1,3-thiazol-5-yl]-4-phenyl-1H-imidazol-1-yl}propanoic acid
4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(2-phenoxyethyl)acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(2,5-dioxoimidazolidin-4-yl)propanamide
4-{[3-(4-cyclopropanecarbonylphenyl)phenyl]methyl}morpholine
4-[(5-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
(3S,4S)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-[2-(4-fluorophenyl)ethyl]-2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]acetamide
6-ethoxy-3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-(2-benzamido-5-methylphenyl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(3-fluoropyridin-4-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-[(4-methoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)acetamide
N-benzyl-2-{4-[4-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}acetamide
3-methyl-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
4-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
N-{[1-(2-amino-6-methoxypyrimidin-4-yl)piperidin-3-yl]methyl}acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)piperidin-2-one
3-(1-methyl-1H-1,2,4-triazol-3-yl)-1-(thiophen-3-ylmethyl)urea
5-methanesulfonyl-1'-(pyridin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]