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4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[3-(pyridin-3-yl)propyl]acetamide
N3-benzyl-1-cyclopropyl-N5-[(2-methoxynaphthalen-1-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-ethyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
3-(pentan-2-yl)-8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1'-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-(difluoromethyl)-4-(3,5-dimethoxyphenyl)-3-methyl-1H-pyrazole
1-methyl-4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
2-{[1-cyclohexyl-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
[3-(hydroxymethyl)-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-yl]methanol
2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-5-(dimethylamino)-2,3-dihydropyridazin-3-one
2-(5-methyl-1,2-oxazol-3-yl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(pyrazin-2-yl)piperidin-4-yl]oxy}benzamide
3-acetyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
(4aS,7aR)-1-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-2-oxoethyl}acetamide
N-(3-fluorophenyl)-4-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)benzamide
2-(furan-3-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
2-({6-[(E)-2-cyclohexylethenyl]pyrimidin-4-yl}amino)ethan-1-ol
1-({3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-3,5-dimethyl-1H-pyrazole
3-[(2R,3R,6R)-5-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
9-[2-(3,4-dimethylphenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-{[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]amino}pentan-2-ol
{5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]furan-2-yl}methanol
2-(1-cyclopentyl-4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperazin-2-yl)ethan-1-ol
4-[5-(4-methoxyphenyl)furan-2-carbonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
2-(phenylamino)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-5-carboxamide
1-{[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
3-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-ethyl-4-methyl-5-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}-1,3-thiazol-2-amine
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(furan-2-yl)ethyl]propanamide
8-[(4-methoxyphenyl)methyl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(1H-indazole-3-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-propoxypropan-1-one
(2S)-2-acetamido-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
2-(cyclopropylamino)-1-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
(1r,4r)-4-{[2-(dimethylamino)-2-(4-methylphenyl)acetamido]methyl}cyclohexane-1-carboxylic acid
3-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylpropanamide
(4S,6R)-N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-({5-[(2,5-dichlorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
6-(3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-3-oxopropyl)-2,3,4,5-tetrahydropyridazin-3-one
methyl 4-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
N-[(2-ethylpyrimidin-4-yl)methyl]-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
N-cyclopropyl-6-[3-(1-methoxyethyl)phenyl]pyridazin-3-amine
2-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}pyrimidine-5-carboxylic acid
N-[(3-chlorophenyl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide