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4-ethyl-5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
7-[2-(1H-pyrazol-1-yl)butanoyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]acetamide
N-[(3R,4R)-1-(3-cyano-4,6-dimethylpyridin-2-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}(pyridin-2-yl)methanol
3-cyclohexyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-({[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}methyl)piperidin-3-ol
2-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,4-dihydroquinolin-4-one
N-[3-(3-chlorophenyl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
methyl 2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)acetate
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-(1H-imidazol-2-ylmethyl)-4-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-1,4-diazepane-6-carboxylic acid
(1R,3S,5S)-8-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-8-azabicyclo[3.2.1]octan-3-ol
2-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(1-ethylpiperidin-4-yl)-N-(2-methoxyethyl)acetamide
3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-ol
2-(2-methyl-6-{spiro[indene-1,4'-piperidine]-1'-yl}pyrimidin-4-yl)ethan-1-amine
N-(3-chloro-2-ethoxyphenyl)-2-methyl-3-oxo-4-phenylpiperazine-1-carboxamide
5-methanesulfonyl-2-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidin-4-amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)piperidin-2-one
1-[4-(2,3-dihydro-1-benzofuran-5-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
2-amino-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyridine-4-carboxamide
8-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-8-azaspiro[4.5]decane-7,9-dione
1-(5-methylpyridin-3-yl)-3-[(4-phenyloxan-4-yl)methyl]urea
N2-benzyl-6-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]-1,3,5-triazine-2,4-diamine
N-benzyl[(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)amino]sulfonamide
3-(5-methyl-1,2,4-oxadiazol-3-yl)-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidine
3-hexyl-8-(pyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-4-(4-methylphenyl)-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidin-3-yl]acetamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-hydroxyphenyl)ethan-1-one
(2S,4R)-4-amino-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
2-[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
5-amino-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide
3-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(methyl)amino)methyl]phenol
2-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]pyridine-4-carbonitrile
[(3R,4R)-1-(7,8-dimethylquinolin-4-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-(2-chloro-6-methylphenyl)-1H-1,3-benzodiazole-5-carbonitrile
1-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2,4,6-trifluorophenyl)ethan-1-one
5-({methyl[(3-{2-[4-(naphthalene-1-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
1-{4-[1-(2,3-dihydro-1H-inden-5-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
3-{4-[1-(methoxymethyl)cyclopropanecarbonyl]piperazin-1-yl}phenol
2-(2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-indazol-3-one
4-({5-[(oxan-2-ylmethyl)sulfanyl]-4-phenyl-4H-1,2,4-triazol-3-yl}methyl)piperidine
2-amino-4-[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]quinazoline-6-carboxylic acid
2-methyl-N-({3-methyl-7-[(2E)-2-methylbut-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-3-carboxamide
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N'-(2,5-dimethoxyphenyl)propanediamide