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5-(4-fluoropiperidin-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(2H-1,2,3-benzotriazol-2-yl)-N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]acetamide
1-[4-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
1-(2-methoxyacetyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
4-hydroxy-N,2-dimethyl-N-[1-(pyridin-3-yl)pentyl]pyrimidine-5-carboxamide
(3aS,6aS)-N-[2-(2-fluorophenoxy)pyridin-3-yl]-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-(1,2-oxazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-methyl-4-(morpholin-4-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]propan-1-one
4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-2,6-dimethoxyphenol
N-{2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)formamido]ethyl}pyridine-3-carboxamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-({5-[(2,6-difluoro-3-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-(5,6-dimethylpyridine-3-carbonyl)-3-phenylpiperazine
[(3R,5R)-1-[4-(difluoromethoxy)benzoyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
4-chloro-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylbenzene-1-sulfonamide
butyl N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}carbamate
2-{4-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]phenoxy}acetamide
3-[1-(4-methylphenyl)cyclopentyl]-5-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,2,4-oxadiazole
(2R,3R,6R)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
4-amino-N-{1-[(4-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}azepane-1-carboxamide
(1R,3S)-7-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
[(2-chloro-3,4-dimethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
1-(furan-3-carbonyl)-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3S,4S)-N-(2-fluoropyridin-3-yl)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
1-[4-methyl-2-({[4-(3-methylpiperidin-1-yl)phenyl]methyl}amino)pyrimidin-5-yl]ethan-1-one
3-{[1-(4-methoxyphenyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
8-methyl-2-propyl-N-[2-(pyridin-3-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-({[3-(1H-imidazol-2-yl)phenyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-[(1S,5R)-3-[2-(3,4-dimethylphenyl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-{[4-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazin-1-yl]methyl}piperidin-3-ol
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(methylamino)ethyl]amino}methyl)piperidin-2-one
1-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-4-(4-methoxyphenyl)butan-1-one
2-(2-methoxyethyl)-9-[3-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-fluoro-6-{[(2-methoxyethyl)[(4-methylphenyl)methyl]amino]methyl}phenol
2,6-dimethyl-4-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]quinoline
3-[3-(methylsulfamoyl)phenyl]-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
(cyclopropylmethyl)({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
(3R,4R)-4-ethyl-1-(2-methoxypyridine-3-carbonyl)piperidine-3,4-diol
{5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]furan-2-yl}methanol
3-(3-methoxypiperidine-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
2-methyl-6-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-(3-chlorophenyl)-5-methyl-4-[2-(2-oxopyrrolidin-1-yl)acetyl]piperazin-2-one
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]-N-methylbenzamide
ethyl (4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
3-[1-(6-hydroxypyridine-3-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one