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1-(4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)ethan-1-one
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrazin-2-amine
3-ethyl-6-(1,4-oxazepane-4-carbonyl)-3H-imidazo[4,5-b]pyridin-2-amine
(4aS,7aR)-1-[(3-ethoxyphenyl)methyl]-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[4-(2-fluorophenoxy)phenyl]-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidine-4-carboxamide
(4aS,7aR)-1-(1,2-oxazole-3-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-chloro-N-[(3S,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-4-hydroxyquinoline-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}propanamide
{[4-(3-fluorophenyl)oxan-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-(2-hydroxyethyl)-2-(morpholin-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-5-carboxamide
6-chloro-N,N-dimethyl-3-({[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
1-benzyl-N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-amine
(4aS,7aR)-1-[2-(5-acetylthiophen-3-yl)acetyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-butyl-8-[4-(propan-2-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-N-[1-(1H-indol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2S)-2-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}-3-(pyridin-4-yl)propanoic acid
4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2,6-dimethylquinoline
N-[(5,6-dimethylpyridin-3-yl)methyl]-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[(4-fluorophenyl)methyl]propanamide
4-{3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-ethoxy-N-[(1-ethylpyrrolidin-3-yl)methyl]-5-methylbenzene-1-sulfonamide
4-[(dimethylamino)methyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}azepan-4-ol
ethyl 4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine-1-carboxylate
3-{[(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}-4H-chromen-4-one
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2,5-dimethoxybenzene-1-sulfonamide
(2S,3S)-2-amino-N-[(3-chlorophenyl)methyl]-3-methyl-N-propylpentanamide
N,N-dimethyl-7-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}pyridine
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-indole-6-carboxamide
4-(4-ethyl-5-methylpyrimidin-2-yl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-[2-(1H-imidazol-1-yl)ethyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(4aR,7aS)-1-methanesulfonyl-4-(4-methoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-({[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}methyl)phenyl]butanamide
1,1-dioxo-N-[4-(thiophen-2-ylmethoxy)phenyl]-1λ6-thiomorpholine-4-carboxamide
7-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-[(3-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
(1S,4S)-2-(3-chlorophenyl)-5-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
4-{[2-(3-hydroxypiperidin-1-yl)-6-methylquinolin-3-yl]methyl}-1-methylpiperazin-2-one
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinazolin-4-amine
1-benzyl-4-(pyridin-4-yl)-1,4-diazepan-6-ol
5-(4-ethoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N2-[(1-benzylpiperidin-4-yl)methyl]-N2-methylpyrimidine-2,4-diamine