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3-(3-chlorophenyl)-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidine
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[2-methyl-4-(pyrrolidine-1-carbonyl)phenyl]urea
2-[({5-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)sulfanyl]pyrimidine
methyl 2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-3-carboxylate
3-phenyl-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
(2E)-3-(3-chlorophenyl)-1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}prop-2-en-1-one
4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]-1-(thian-4-yl)piperidine
3-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indazole
N-methyl-N-[2-(pyridin-2-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[(dimethylamino)methyl]-1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-3-ol
3-(1-methyl-1H-imidazol-4-yl)-5-[3-(1H-pyrazol-4-yl)propyl]-1,2,4-oxadiazole
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
8-(oxolane-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-cyclohexanecarbonyl-N-[2-(2,3-dimethoxyphenyl)ethyl]pyrrolidine-2-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
methyl 4-(4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)benzoate
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1-ethyl-5-oxopyrrolidin-3-yl)benzamide
N-[2-(dimethylamino)ethyl]-3-{[(4-methylphenyl)methyl]amino}benzamide
4-oxo-4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butanamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
N-(2,2-difluoroethyl)-4-{[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}benzamide
2-(5-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-[2-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
N'-(5-chloro-2-methylphenyl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]propanediamide
N-[3-(cyclohexylsulfanyl)propyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-methyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine
2-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}quinolin-8-ol
N-(oxan-4-ylmethyl)-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(pyridin-4-yl)piperazine
8-(4-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-(aminomethyl)-2-(2-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1H-imidazole-2-carboxamide
4-[(5-methoxy-1H-indazol-3-yl)methyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
2-methoxy-1-{1'-[2-(pyrrolidin-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-[(3R,4S)-1-(4-chlorobenzoyl)-4-cyclopropylpyrrolidin-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-(1-methyl-1H-pyrazol-4-yl)-4-[3-(trifluoromethyl)piperidine-1-carbonyl]quinoline
1-(1H-pyrazol-3-ylmethyl)-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
1-benzyl-N3-cyclohexyl-N5-ethyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-methyl-2-[4-(5-methylpyrazine-2-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
2-[(2,3-dimethoxyphenyl)methyl]-4-{4-[(2S)-2-hydroxy-2-phenylacetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 3-benzyl-1-methanesulfonylpiperidine-3-carboxylate
4-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
4-chloro-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
methyl 1-{[7-(methylsulfanyl)-2-oxo-1,2-dihydroquinolin-3-yl]methyl}piperidine-2-carboxylate
4-[1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-3-yl]benzoic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4,4,4-trifluorobutanamide
(2S,4R)-N-ethyl-4-(3-fluorobenzamido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
5-ethyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine