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4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]pyrimidine
5-ethyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-cyclopropyl-1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-{[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl)amino}propane-1,2-diol
2-(3-hydroxyadamantan-1-yl)-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
4-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]morpholine
1-tert-butyl-4-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}pyrrolidin-2-one
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(2R,6S)-1-(1H-imidazole-2-carbonyl)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
4-(1H-pyrazol-1-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
4-{[3-(acetamidomethyl)piperidin-1-yl]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
N4-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-6-methylpyrimidine-2,4-diamine
1-[(3-chloro-2,6-difluorophenyl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
2-[8-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
2-{2-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]ethyl}pyridine
1-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-4-[(2-methylphenyl)methyl]piperazine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-hydroxypropyl)piperidine-4-carboxamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
1-(5-tert-butyl-2-methoxyphenyl)-3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]urea
1-[({5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}carbamoyl)methyl]piperidine-4-carboxamide
N-[(3-methylthiophen-2-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
5-[2-(4-methylphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2-{[7-(5-cyanopyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)acetamide
1-methyl-5-{1-methyl-octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1H-1,2,3-benzotriazole
N-(1H-imidazol-2-ylmethyl)-N,6-dimethyl-2-phenylpyrimidin-4-amine
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperazine
1-cyclopentyl-N3-(1,2-diphenylethyl)-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(4-benzylpiperazin-1-yl)ethyl]-6-cyclopropylpyrimidin-4-amine
9-(furan-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-methylphenyl)-N-{2-[2-(pyrimidin-2-ylsulfanyl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
1-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-{2-[({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)methyl]phenoxy}ethan-1-ol
(4aS,7aR)-1-(5-acetylthiophene-2-carbonyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(benzenesulfonyl)-1-[2-(furan-2-yl)azepan-1-yl]propan-1-one
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-[2-(pyridin-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[2-(2-methoxyethyl)morpholine-4-carbonyl]-2-phenylpyrimidin-4-ol
(3aR,6aR)-2-cyclopentanecarbonyl-5-(4-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{2-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-cyclopentylpiperazine
1-methyl-4-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-3-phenyl-1H-pyrazole
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methyl-2-(methylamino)propan-1-one
7-[(2-fluorophenyl)methyl]-2-(5-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-(2-methoxyphenyl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazole-4-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]propanamide
1-[(5-cyclopentylthiophen-2-yl)methyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
1-{[4-(dimethylamino)-1-ethylpiperidin-4-yl]methyl}-3-(3-fluoro-5-methylphenyl)urea
N-(2-{[(6,8-dimethyl-2-oxo-2H-chromen-4-yl)methyl]amino}ethyl)pyridine-3-carboxamide
3-({[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}(methyl)amino)propane-1,2-diol
N,3-dimethyl-5-propyl-N-[3-(1H-pyrazol-1-yl)propyl]-1-benzofuran-2-carboxamide