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1-benzyl-N3-[2-(3-chlorophenyl)ethyl]-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
9-(2-amino-6-methylpyrimidin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1,2-oxazole-3-carbonyl]-1-ethyl-3-methylpiperazin-2-one
1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
2-amino-7-methyl-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-5H,7H-thieno[3,4-b]pyridine-3-carbonitrile
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methoxy-N-{4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}acetamide
(3E)-N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbut-3-enamide
6-methyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine-3-carbonitrile
1-{1-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(3aS,6aS)-5-(1-benzoxepine-4-carbonyl)-1-methyl-octahydropyrrolo[3,4-b]pyrrole
2-(2-{1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-{8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
11-({[3-fluoro-5-(trifluoromethyl)phenyl]methyl}amino)-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N5-cyclopropyl-N6-[2-(2-methoxyphenyl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(3S)-3-ethyl-4-(1-propyl-1H-pyrazole-5-carbonyl)morpholine
2-(4-{6-[(2-hydroxyethyl)(methyl)amino]pyridazin-3-yl}phenyl)-2-methylpropanenitrile
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-amino-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
3-{methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}propane-1,2-diol
(2E)-N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-3-(1H-imidazol-4-yl)prop-2-enamide
N-methyl-5-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
(1R,5S,6S)-N-(2,3-dihydro-1H-inden-2-yl)-3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
4-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine
8-chloro-2-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}quinoline
1-[(2-methylfuran-3-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethoxy)ethan-1-ol
3-chloro-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylbenzene-1-sulfonamide
1-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
N-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-2-[4-(6-methoxypyridin-2-yl)-1H-pyrazol-1-yl]acetamide
4-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
methyl 2-oxo-8-[(2E)-3-phenylprop-2-en-1-yl]-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(2-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,3S,5S)-3-(4-methoxyphenyl)-8-[3-(1H-pyrazol-1-yl)benzoyl]-8-azabicyclo[3.2.1]octane
6-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-5,6,7,8-tetrahydro-1,6-naphthyridine
4-(3-methylpyridine-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-1-phenyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(1-phenylcyclopentyl)methyl]acetamide
3-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
(1S,5R)-6-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-(3-fluorophenoxy)-1-[3-(methylcarbamoyl)pyridin-2-yl]piperidine-4-carboxylic acid
(1S,6R)-N-(3-methoxyphenyl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-thiazole
N,N,2-trimethyl-4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-sulfonamide
propan-2-yl 4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carboxylate
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-[2-(2-fluorophenoxy)ethyl]-3-azaspiro[5.5]undecan-9-amine
3-(aminomethyl)-4-(2-phenylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one