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1-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-methoxypiperidine
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-ethyl-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidin-4-amine
2-(4-{[3-(aminomethyl)piperidin-1-yl]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one
8-fluoro-3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(propane-2-sulfonyl)piperidin-3-amine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
4-(6-methoxypyrimidin-4-yl)-2-(trifluoromethyl)morpholine
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-chlorobenzamide
N-phenyl-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]pyrimidin-2-amine
2-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}quinoxaline
2-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1-benzofuran-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propan-1-one
2,3-dimethyl-7-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-4-propylpyrimidine
1-(3-phenylpropyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-{[4-(2-phenylazetidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}-1H-1,3-benzodiazole
4-{5-[1-(furan-2-ylmethyl)piperidin-3-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
ethyl 1-(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazole-4-carbonyl)piperidine-4-carboxylate
N-(2-{7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
1-tert-butyl-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(thiophen-2-yl)ethan-1-one
2-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}-8-methoxyquinoline
ethyl 3-[(2-methylphenyl)methyl]-1-(3-methylthiophene-2-carbonyl)piperidine-3-carboxylate
N4-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
4-[3-ethoxy-4-methoxy-5-(prop-2-en-1-yl)phenyl]-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
2-[1-(4-chlorophenyl)cyclobutyl]-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(trifluoromethyl)benzamide
3-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}azetidin-3-yl)pyridine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-(1-{1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
4,6-dimethyl-2-oxo-N-[3-(pyridin-3-yloxy)propyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-phenylacetamide
3-{2-[2-(2-methoxyethyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-N-methylbenzamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
3-({[1-(furan-2-carbonyl)piperidin-3-yl]carbamoyl}amino)-N,4-dimethylbenzamide
(2S)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-methylbutanamide
2-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-4-(1H-pyrrol-1-yl)phenol
[(3R,4R)-1-(2,6-dimethoxybenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-[3-(2-ethylpiperidine-1-carbonyl)phenyl]cyclopentanecarboxamide
6-[(1-ethyl-1H-indazol-3-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-methyl-6-(1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
6-(1-benzofuran-2-ylmethyl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-[(phenylsulfanyl)methyl]furan-2-carboxamide
6-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}-1-methyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
N1-(pyridin-3-yl)-N3-{1H-pyrrolo[2,3-b]pyridin-6-yl}propane-1,3-diamine
1-{4-[6-hydroxy-4-(1-methyl-1H-imidazole-4-carbonyl)-1,4-diazepan-1-yl]piperidin-1-yl}ethan-1-one
(2S,4S)-4-amino-N-methyl-1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide