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N-ethyl-1-(2-methylpropyl)-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}-2-(2-phenylethyl)piperidine
(3R,4R)-1-[(4-chloro-3-fluorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(4-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-2-chloro-6-methoxyphenoxy)acetamide
2-[3-(1-methoxyethyl)phenyl]-3-(piperidine-1-carbonyl)pyridine
4-{4-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-4-carboxamide
N-cyclopentyl-5-[2-(5,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(3-chlorophenyl)-4-{[(1s,4s)-4-aminocyclohexyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-ethyl-4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyridin-2-one
2-(2-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-[(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
1-methyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(pentan-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-chloro-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylbenzamide
2-[2,4-dichloro-3-(pyrrolidin-1-ylmethyl)phenoxy]-3-methoxypyrazine
2-(pyridin-4-ylsulfanyl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethan-1-one
2-[1-methyl-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-(1-{[1-(prop-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}piperidin-3-yl)furan-2-carboxamide
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(2-propoxypropyl)acetamide
2-amino-4-(5-ethylfuran-2-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-(propan-2-yl)-2-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
5-amino-3-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1H-indazole
4-{[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}-1-(propan-2-yl)pyrrolidin-2-one
N-(2-{5-[1-(furan-2-carbonyl)piperidin-2-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)acetamide
4-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
2-(2,4-difluorophenyl)-2-[2-(1-ethylpiperidin-4-yl)acetamido]acetic acid
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(3,5-dimethylphenyl)piperazin-2-one
1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
6-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}pyridine-3-carbonitrile
3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-1-(2-methoxy-6-methylphenyl)urea
(5S,9aS,9bS)-2-phenyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenyl]-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(3-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-N-{[3-methyl-7-(3-phenoxypropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-3-carboxamide
2-[2-({4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenoxy]acetic acid
{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
2-{4-[3-methoxy-5-(trifluoromethyl)phenyl]phenyl}-N,N-dimethylacetamide
2-cyclopropyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
2-(morpholin-3-yl)-1-[4-(naphthalen-1-yl)piperazin-1-yl]ethan-1-one
2-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1-benzofuran-5-carboxamide
2-[2-(methylamino)pyridine-4-carbonyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
6-methyl-N4-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)pyrimidine-2,4-diamine
methyl 4-(7-fluoro-2-methylquinoline-4-carbonyl)piperazine-1-carboxylate