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N4-{3-[cyclopentyl(methyl)amino]propyl}-6-methylpyrimidine-2,4-diamine
{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
5-cyclopropyl-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,3,4-oxadiazol-2-amine
4-(cyclopropylamino)-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-({1-[(2-hydroxynaphthalen-1-yl)methyl]piperidin-3-yl}methyl)acetamide
phenyl({1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl})methanol
2-methyl-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2-ethoxyethyl)-5-[3-(piperidin-1-yl)azetidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-1,4-diazepane
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
3-[1-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)piperidin-4-yl]-1,3-oxazolidin-2-one
1'-(5-methyl-1,3-oxazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-methyl-6-[3-(1H-pyrazol-5-yl)phenyl]pyridazine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-(2-phenoxyethyl)-8-(1,3-thiazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]acetamide
2-[4-(4-chloro-2-hydroxybenzoyl)-2-oxopiperazin-1-yl]benzonitrile
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}thiomorpholine
2-cyclopropyl-4-hydroxy-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
5-[(3S)-3-ethylmorpholine-4-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
1-{2-[(1E)-pent-1-en-1-yl]pyrimidin-4-yl}piperidin-3-ol
6-fluoro-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[1-(carbamoylmethyl)piperidin-4-yl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(oxan-3-ylmethyl)acetamide
[(3R,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(2-phenoxyethyl)benzamide
1-(2-methoxyphenyl)-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine
{2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}urea
N-[2-(morpholin-4-yl)ethyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N,1-dimethyl-2-oxo-N-[1-(pyridin-3-yl)pentyl]-1,2-dihydropyridine-3-carboxamide
(2S)-N-[3-(4-fluorophenyl)phenyl]-1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]pyrrolidine-2-carboxamide
N,N-dimethyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-sulfonamide
7-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1H-pyrazol-3-yl]phenol
N-[4-methyl-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][1-(2-methoxyphenyl)ethyl]methylamine
[(6-chloropyridin-3-yl)methyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]propane-1,3-diol
3-{5-[(4-ethyl-1,4-diazepan-1-yl)methyl]thiophen-2-yl}prop-2-yn-1-ol
N-[2-(azepan-1-yl)ethyl]-2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-(propan-2-yl)acetamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-fluoro-2-methylphenyl)ethan-1-one
2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]acetic acid
4-(2-methyloxolane-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2-methoxyethyl)-3-(oxolan-2-ylmethyl)-1-(2-phenylphenyl)urea
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methoxyphenyl)methyl]piperidine
1-[3-(4-chlorophenyl)-3-phenylpropanoyl]-1,4-diazepan-5-one
N-(1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-1H-pyrazole-4-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine