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2,5-dimethyl-N-(oxolan-2-ylmethyl)-N-(3-phenylprop-2-yn-1-yl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-5-(piperidin-1-ylmethyl)pyridine
N-{[4-methoxy-3-(pyridin-3-ylmethoxy)phenyl]methyl}-2,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1H-indole-7-carboxamide
3-(4-tert-butylbenzoyl)-1-ethylpiperidine
4-[6-(piperidin-1-yl)pyrimidin-4-yl]-2-(trifluoromethyl)morpholine
N-methyl-2-(oxolan-2-ylmethoxy)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-methylpropyl 4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carboxylate
3-(2-amino-1,3-thiazol-4-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propan-1-one
3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-[2-(dimethylamino)ethyl]-4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-cyclopropylacetamide
N-[(1-cycloheptylpiperidin-3-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(4aS,7aR)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-3-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)pyridin-2-amine
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propylpyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
(3S,4R)-1-[(5-chlorothiophen-2-yl)methyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
ethyl 1-(2-fluorobenzenesulfonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-(2-methylpropyl)-1,4-diazepan-5-one
8-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(furan-2-ylmethyl)-4-methyl-N-(3-methylbutan-2-yl)pyridine-3-carboxamide
6-(isoquinolin-5-yl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
2-(3-fluoro-4-hydroxyphenyl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
6-methoxy-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}pyrimidin-4-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-methylpiperidin-2-one
methyl 3-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-methyl-5-{[methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]methyl}pyrimidin-2-amine
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(3-methoxypropyl)piperidine-3-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[4-(pyridin-2-yl)butyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)pyrimidine-5-carboxamide
1-(cyclobutylmethyl)-3-hydroxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
1-(3-chlorophenyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
6-{4-[(5-methylnaphthalen-1-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
2-[4-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]pyridine
(2S)-2-{[5-methyl-2-(2-methylpropanamido)phenyl]formamido}-3-phenylpropanamide
methyl[(4-{2-[1-(pyridine-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
N-(1-ethyl-1H-pyrazol-5-yl)-2-{4-[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrazol-1-yl}acetamide
(2E)-1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyridin-2-yl)prop-2-en-1-one
N-methyl-N-{3-oxo-3-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propyl}methanesulfonamide
N-benzyl-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-phenyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
[(3R,4R)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
2-methyl-8-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(oxolan-3-yl)-5-(2-phenoxypropan-2-yl)-1,2,4-oxadiazole
2-[(2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
2-(2-chloro-6-methoxyphenyl)-2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}acetic acid
N-(3-{[({4-[methyl(phenyl)amino]phenyl}methyl)amino]methyl}-5-(pyrrolidine-1-carbonyl)phenyl)acetamide