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4-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-3-yl}acetamide
1-(3,5-dimethylphenyl)-4-(2-methylpyridin-4-yl)piperazin-2-one
6-ethyl-3-(2-methoxyethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(4-methylphenoxymethyl)piperidine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[2-(1H-imidazol-4-yl)ethyl]piperidine-3,5-dicarboxamide
{1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
4-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1λ6-thiane-1,1-dione
2-{[4-(2-methoxyphenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-[(5-methylpyrazin-2-yl)methyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
(furan-3-ylmethyl)(methyl){[5-(propane-2-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
(3S,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
2-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[2-(4-methoxyphenyl)phenyl]-1-propylpyrrolidine-2-carboxamide
2-(4-methoxyphenyl)-N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)acetamide
4-[(2-fluorophenyl)methyl]-1-(4-methoxyphenyl)piperazin-2-one
(3S,4S)-4-(4-fluorophenyl)-1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-3-ol
N-[4-(2-fluorophenoxy)phenyl]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxamide
5-{1-[(2,5-dimethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(1,4-dioxan-2-ylmethyl)-1-benzofuran-2-carboxamide
3-[1-(5-phenylpentanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
2-(1H-1,2,3-benzotriazole-5-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
8-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[4-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
2-[2-(quinolin-3-yl)phenyl]ethan-1-amine
2-ethyl-5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}pyrimidine
2-{4-cyclopentyl-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
6-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-5,6,7,8-tetrahydro-1,6-naphthyridine
4-[4-(4-chlorophenyl)-4H-1,2,4-triazol-3-yl]-2-methoxyphenol
4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-1-(thiophene-2-carbonyl)piperidine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidin-2-one
4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
3-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2,3-dihydro-1,3-benzoxazol-2-one
[1-(3-phenylpropyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
5-(3-cyclopropyl-1H-pyrazol-5-yl)-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-{4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-6-methoxypyrimidin-4-amine
2-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}benzoic acid
4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-cyclopentylpyrrolidin-2-one
4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-[benzyl(methyl)amino]-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]ethan-1-one
5-{[(5-chlorothiophen-2-yl)methyl]amino}-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
1-(3-methylpiperidin-1-yl)-3-[3-(piperidin-1-yl)azetidin-1-yl]propan-1-one
4-[5-(thiomorpholine-4-carbonyl)-1H-pyrazol-3-yl]phenol
2-[(3-chlorophenyl)methyl]-N-methyl-N-(pyridin-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-cyclohexyl-3-({[(2-fluoro-4-methylphenyl)carbamoyl]methyl}amino)propanamide