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2-cyclopropyl-5-(3,3-diphenylpiperidine-1-carbonyl)pyrimidine
6-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
3-[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
(1S,5R)-6-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-6-(1H-pyrazol-4-yl)quinoline
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(6-oxo-1,6-dihydropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-methyl-5-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4R)-1-benzyl-4-({[4-(benzyloxy)phenyl]methyl}amino)-N-methylpyrrolidine-2-carboxamide
methyl (2R,4S)-1-[2-(2-chloro-5-methylphenoxy)-2-methylpropanoyl]-4-hydroxypiperidine-2-carboxylate
1-[4-(4-aminopyrimidin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-{imidazo[1,2-a]pyridin-3-yl}ethan-1-one
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(thiophen-2-yl)propan-2-yl]butanamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-2-(morpholin-4-yl)benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-methoxybenzamide
2-hydroxy-1-[3-(pyridin-3-yl)azetidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
methyl[(1-methylpiperidin-3-yl)methyl][(2,3,4-trimethoxyphenyl)methyl]amine
1-[2-amino-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-(2-methoxyethyl)-4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-ol
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
5-methyl-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-carboxamide
2-({2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-5-methyl-1,3,4-thiadiazole
1-cyclopropanecarbonyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[4-(3-methoxyphenyl)phenyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-3-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-methyl-4-phenyl-3-[1-(pyridine-4-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,5S)-1-benzyl-N-[(4-phenylphenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
6-[1-(2,3-dihydro-1H-inden-4-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
(4aS,8aR)-6-(2-amino-4-methylpyrimidine-5-carbonyl)-1-butyl-decahydro-1,6-naphthyridin-2-one
(3R)-3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
4-[3,5-dichloro-4-(propan-2-yloxy)phenyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-butyl-6-methyl-2-(4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-2-carbonitrile
3-{[(6-chloro-2H-chromen-3-yl)methyl](methyl)amino}-N-methylbutanamide
6,7-dimethoxy-2-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
4-(2,3-dihydro-1H-inden-5-yloxy)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
8-fluoro-2-{[(oxan-3-ylmethyl)amino]methyl}quinolin-4-ol
2-{5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-(2-chloro-4-{[2-(ethoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclopropane-1-carboxamide
N-ethyl-5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
N-(2-hydroxyethyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(3S,4R)-1-(5-ethyl-1,3,4-thiadiazol-2-yl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(morpholine-4-carbonyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzene-1-sulfonamide
5-{2-[(5-cyclopropyl-1,3,4-thiadiazol-2-yl)carbamoyl]ethyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide