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N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-[2-(dimethylamino)ethyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
3-({[(2-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
2-{3,5-dimethyl-4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-1H-pyrazol-1-yl}ethan-1-ol
[2-(3-fluorophenyl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
N-benzyl-5-[ethyl(pyridin-4-ylmethyl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
3-[2,4-bis(hydroxymethyl)phenyl]-5-[2-(piperidin-2-yl)ethyl]phenol
methyl 1-[(3R,5S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[1-(1H-imidazol-1-yl)butan-2-yl]pyrazolo[1,5-a]pyridine-3-carboxamide
2-[1-butyl-5-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-[(3-chlorophenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-{2-[2-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
N-[3-(2-chlorophenoxy)propyl]-N-methyloxolane-3-carboxamide
(1R,2S)-2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}cyclopentane-1-carboxamide
N,N-dimethyl-3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxamide
[1-(4-methoxyphenyl)ethyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,3-benzothiazole-5-carboxamide
2-[1-cyclohexyl-4-(1H-indol-2-ylmethyl)piperazin-2-yl]ethan-1-ol
(1R,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
[(3-fluoro-4-methoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
2-[4-(3,6-dimethylpyrazin-2-yl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
6-[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]quinoxaline
6-[(diethylamino)methyl]-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,2R)-N1-butyl-N1-[(4-fluorophenyl)methyl]-N2-methylcyclohexane-1,2-dicarboxamide
4-{4-[1-(piperidin-1-yl)ethyl]phenyl}thiophene-2-carboxamide
2-(4-phenyl-1H-imidazol-5-yl)benzoic acid
2-ethyl-7-methoxy-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-benzyl-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
methyl 3-{[4-(methylsulfanyl)phenyl]methyl}-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S)-N-(6-methoxy-2H-1,3-benzodioxol-5-yl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
2,7-dimethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2-hydroxyethyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-2-carboxamide
7-(2,5-difluorobenzoyl)-N4-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-[(3,5-difluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-methyl-2-oxo-N,N-bis(pyridin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
6-[2-(4-chlorophenyl)morpholin-4-yl]-N-ethyl-N-methylpyridine-3-carboxamide
7-[2-(cyclohex-1-en-1-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
3-[ethyl({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)amino]-1λ6-thiolane-1,1-dione
1-(2-methyl-5-sulfamoylphenyl)-3-[2-(pyrrolidin-1-yl)ethyl]urea
N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methylpropanamide