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8-(1H-1,2,3-benzotriazole-5-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-({5-cyclopropyl-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
4-(dimethyl-1,3-oxazole-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,9aR)-3-methyl-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]acetamide
N,N-dimethyl-3-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)benzamide
2-amino-3-ethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-2-phenylmorpholine
3-(4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)propanoic acid
N-methyl-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}thiophene-2-carboxamide
2-[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
1-{[1-(6-{[3-(dimethylamino)propyl]amino}pyridine-3-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
3-[methyl({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amino]propane-1,2-diol
3-(2-chlorophenyl)-1-(1,4-diazepan-1-yl)-3-phenylpropan-1-one
1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-N-methylfuran-2-carboxamide
1-[(3-methylphenyl)methyl]-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazine
4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
[(4-methoxynaphthalen-1-yl)methyl](methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
6-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methylbenzamide
2-{4-[(2,3-difluoro-6-methoxyphenyl)methyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]amine
4-methoxy-N-(2-methoxyethyl)-2-({1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-(1-cycloheptylpiperidin-3-yl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
5-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-(3,4,5-trifluorophenyl)urea
2-(3-methoxypropyl)-9-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
benzyl({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2-phenylethyl)amine
2,2-difluoro-N-[1-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)propan-2-yl]-2H-1,3-benzodioxole-5-carboxamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxyethan-1-one
(4aR,7aS)-1-propanoyl-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[(5-phenyl-1H-pyrazol-3-yl)methyl]amine
6-fluoro-2-({[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino}methyl)quinolin-4-ol
3-{1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}benzoic acid
1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-4-(1H-pyrazol-3-yl)piperidine
3-[3-cyclopropyl-5-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
2-methoxy-1-{3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
N-(3-ethoxy-2-hydroxypropyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(3-{[4-(methylamino)pyrimidin-2-yl]amino}propyl)piperidine-4-carboxamide
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[2-(propan-2-yloxy)phenyl]pyridine
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N5-cyclopropyl-N6-[2-(furan-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-phenyl-1-{1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethan-1-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one