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(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-fluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(benzylsulfamoyl)amino]-N-(4-fluoro-2-methylphenyl)acetamide
{[6-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)pyridin-3-yl]methyl}dimethylamine
(7S,9aR)-7-(cyclohexylmethyl)-N-(3-fluorophenyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-methyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-(3-phenoxypropyl)acetamide
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrrolidine-3-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(5-methyl-1,2-oxazol-3-yl)methyl]pyrimidine-5-carboxamide
4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
4-hydroxy-2-(pyridin-3-yl)-N-[(3,4,5-trifluorophenyl)methyl]pyrimidine-5-carboxamide
3-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
3-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
(3aS,6aS)-2-[(6-hydroxynaphthalen-2-yl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}acetamide
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(4-methoxybenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-{1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazol-4-yl}quinolin-4-ol
6-cyclopentyl-N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(1H-1,2,4-triazol-1-yl)propanamide
2-methoxy-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(2S,4S)-4-amino-1-(2,4-difluoro-3-methoxybenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
6-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-(benzyloxy)-8-(2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-{[3-(thiomorpholine-4-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
N-(3-acetamidophenyl)-2-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxamide
1-methyl-4-(quinolin-4-yl)piperazine-2-carboxylic acid
1-[1-(4-benzylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-2-phenylethane-1,2-dione
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carboxamide
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(1H-indol-5-ylmethyl)pyrrolidin-3-yl]methanol
1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(pyridin-2-yl)ethan-1-one
N,1-dimethyl-3-(2-methylpropyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-{3-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}butanamide
5-{[2-(N-methylmethanesulfonamido)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(2-{1-[3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-2-yl}ethyl)acetamide
N-methyl-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
2-[5-(1H-indazol-1-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-(2-hydroxyethyl)-5-[(4-methoxyphenyl)methyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]piperidin-1-yl}acetamide
(3R,4S)-1-(3-chloro-2-methylbenzoyl)-3,4-dimethylpiperidin-4-ol
3-[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]propane-1,2-diol
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-ol
N-(1H-1,3-benzodiazol-2-yl)-2-{[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}acetamide
3-{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}-1,2-benzothiazole
2-methyl-5-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
3-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-1-(4-methylphenyl)urea
1-[2-methoxy-5-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-[(3R,4S)-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-4-(dimethylamino)piperidin-3-yl]propan-1-ol