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N-(3-ethoxypropyl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
5-methyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[3-(1H-imidazol-1-yl)propyl]-1-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)urea
(4aS,7aR)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{[4-(3-propylpyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-ethyl-2-[4-(furan-2-carbonyl)piperazin-1-yl]pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-ethyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2H-1,3-benzodioxole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-ethyl-N-(4-hydroxybutan-2-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-(cyclohexylmethyl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(pyridin-3-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(2-ethoxyethoxy)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
2-[1-(1-methylpiperidin-4-yl)-4-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperazin-2-yl]ethan-1-ol
methyl (2S,4R)-4-(dimethylamino)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-2-carboxylate
2-[1-(1-methoxybutan-2-yl)-4-phenyl-1H-imidazol-5-yl]benzonitrile
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}thiophene-2-carboxamide
2,6-dimethyl-5-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
3,5-difluoro-4-methoxy-N-methyl-N-(pyrazin-2-ylmethyl)benzamide
N-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(3-hydroxyquinoxalin-2-yl)-N-methylpropanamide
3,6-dimethyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrazin-2-amine
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-[5-(3-hydroxyphenyl)pyridin-2-yl]butanamide
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(quinolin-8-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}propanoic acid
N-methyl-3-{[3-(3-phenylpropanoyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
[(3-{2,7-diazaspiro[4.5]decane-7-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)methyl]diethylamine
N'-ethyl-N-(5-methyl-1,2-oxazol-3-yl)-N'-[2-(2-methylphenoxy)ethyl]ethanediamide
2-acetyl-8-[4-(ethylcarbamoyl)pyridin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-2-one
6-butyl-2-{4-[(2-methylpiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
4-{1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
6-[(diethylamino)methyl]-N-[1-(1,3-thiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N1-propyl-N2-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1,2-dicarboxamide
3-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
(2R,3R,6R)-3-(4-methylphenyl)-5-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-(2,4-dimethylphenyl)propyl]acetamide
6-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
(2S,4S)-N-ethyl-4-[(4-ethyl-5-methylpyrimidin-2-yl)amino]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
{[2-methoxy-5-(8-methylquinolin-5-yl)phenyl]methyl}(methyl)amine
2-methyl-6-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
4-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-1-(2-phenylethyl)piperazin-2-one
6-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-amine
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one