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1-(4-chlorophenyl)-5-methyl-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
2-{1-cyclopentyl-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-(5-acetamido-2-methoxyphenyl)-3-(piperidin-1-yl)pyrrolidine-1-carboxamide
2-amino-6-cyclopropanecarbonyl-4-(2-methoxypyrimidin-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(2-fluorophenyl)-N-methyl-1H-pyrazole-5-carboxamide
2-(5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2R,3S,6R)-5-(6-methoxypyrimidin-4-yl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(naphthalene-2-carbonyl)pyrrolidin-3-yl]methanol
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(3-phenylpropyl)-1,4-diazepane
(2S,4S)-4-amino-1-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(4-chlorophenyl)butanamide
N-methyl-N-(2-methylpropyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
2-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]-6-methylpyridine-3-carbonitrile
N-{2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide
6-{1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-({2-[4-(1-methoxyethyl)phenoxy]phenyl}methyl)-4-methylpiperazine
4-[(1R,7S)-4-oxo-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
3-{5-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1'-(1-propyl-1H-pyrazole-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-{4-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperazin-1-yl}phenol
(1S,5R)-6-(cyclobutylmethyl)-3-(2,5-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[3-(4-methoxyphenyl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
2-(cyclohexylmethyl)-N,N-dimethylmorpholine-4-sulfonamide
N-[4-(3-methoxyphenyl)phenyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine-3-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
8-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
2-ethoxy-1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
2-[4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
4-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
9-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
1-(4-{[3-(1H-imidazol-1-yl)propyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-(4-acetyl-4-phenylpiperidine-1-carbonyl)-1-methylimidazolidin-2-one
2-{[2-(dimethylamino)ethyl](methyl)amino}-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
5-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
2-(2,3-dihydro-1H-inden-1-yl)-N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)acetamide
2-[(3,4-dimethoxyphenyl)methyl]-N-(1-methylpyrrolidin-3-yl)-1,3-benzoxazole-6-carboxamide
N-(3-sulfamoylphenyl)-4-(thiophen-2-ylmethyl)piperazine-1-carboxamide
4-(azepane-1-carbonyl)-7-methoxy-2-(1H-pyrazol-4-yl)quinoline
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)cyclobutanecarboxamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
3-(2-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(1H-1,2,4-triazol-5-yl)benzamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyridine-3-carboxamide