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3-acetyl-N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)benzamide
3-({[1-(1-benzothiophene-5-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
5-(3-chloro-5-methylpyridin-2-yl)isoquinoline
N-[(2-fluorophenyl)methyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-ethyl-4-methyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(piperidin-1-yl)propan-1-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(1H-1,2,4-triazol-1-yl)acetamide
2-cyclohexyl-N-methyl-N-(thiophen-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
7-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-1-(1,4-oxazepan-6-ylmethyl)urea
4-(cyclohex-3-en-1-ylmethyl)-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-[(3-chloro-2-fluorophenyl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
3-[N-(propan-2-yl)-1-[4-(trifluoromethyl)phenyl]formamido]propanamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-3,4,7-trimethyl-1H-indole-2-carboxamide
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-methoxypyrimidin-2-amine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3,3,3-trifluoropropan-1-one
methyl 4-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutanoate
(1R,5R)-3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
dimethyl({[4-methyl-5-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
5-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
5-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(2-fluorophenoxymethyl)-1-(furan-3-carbonyl)piperidine
2-[5-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl})amine
N-[(2-methoxyphenyl)methyl]-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-cyclopropyl-3-[({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)sulfamoyl]benzamide
1-(2-methylpropyl)-4-oxo-N-[2-(4-phenylpiperidin-1-yl)ethyl]-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[4-(furan-2-amido)-3-methylphenyl]-5-oxopyrrolidine-3-carboxylic acid
(1R,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(8-fluoroquinoline-2-carbonyl)-1-methylpiperazin-2-one
7-{2-[(4-chlorophenyl)methoxy]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
2-methyl-6-{1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-4-yl}pyrimidin-4-ol
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{3-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-oxo-6-phenyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,2-dihydropyridine-3-carboxamide
1-[3-(2-phenylethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-(cyclopropylmethyl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-({[1-(dimethylcarbamoyl)ethyl](methyl)amino}methyl)benzoic acid
2-{benzyl[1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethan-1-ol
3-acetamido-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-(2-amino-1,3-thiazol-4-yl)-N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]propanamide
1-(azepan-1-yl)-3-{2-methoxy-4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propan-2-ol
N-(4-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}phenyl)acetamide
(2E)-N-cyclopropyl-3-(3-fluorophenyl)-N-{[3-(2-methylpropoxy)phenyl]methyl}prop-2-enamide
7-(3-chlorophenyl)-4-(4-methyl-1H-imidazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
8-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione