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7-(2-methyloxolane-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-(1H-imidazol-4-yl)ethyl]-N-(4-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-phenylpropanamide
9-benzoyl-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
3-chloro-4-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)phenol
(1R,5R)-3-methanesulfonyl-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[(methylcarbamoyl)methyl]sulfamoyl}-N-[2-(pyridin-3-yl)ethyl]benzamide
2-hydroxy-4-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)benzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazine
(3S,4R)-N,N-dimethyl-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-N-(4-methyl-1,3-benzothiazol-2-yl)acetamide
5-({2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
3-[2-(1-methylpiperidin-2-yl)ethyl]-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
1-methyl-8-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-methylpiperazine-2-carboxylic acid
2-[(isoquinolin-5-yloxy)methyl]-N-(2-methoxyethyl)-1,3-oxazole-4-carboxamide
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]benzamide
[5-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-phenyl-1H-imidazol-5-yl)furan-2-yl]methanol
2-(2-chloro-6-methylphenoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2,8-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}quinoline-4-carboxamide
(1R,5R)-6-[(6-fluoroquinolin-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})[2-(4-methylphenoxy)ethyl]amine
N-[4-(4-{[2-(cyclohex-1-en-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
1-{2-[1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
1-{3-[4-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(thiophen-3-ylmethyl)amine
(2S,4S)-4-amino-1-(2-acetamido-1,3-thiazole-5-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
5-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-cyclopentyl-N-[2-(1H-pyrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,2-dihydroquinoxalin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(1H-indol-3-yl)-N-methylpropanamide
(3S,4R)-1-[4-(3-fluorophenyl)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]quinoxaline
2-methyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(2-{4-[(4-ethoxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
6-{[(3,3-diphenylpropyl)amino]methyl}-1,4-oxazepan-6-ol
1-propyl-4-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]amino}pyrrolidin-2-one
3,4-dimethyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-5-sulfamoylbenzamide
1,3-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
5-{[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoxaline
7-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)furan-2-carboxamide
2-{4-[(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-3-methyl-1H-pyrazol-1-yl}ethan-1-ol
N-[(1-{[2-(4-tert-butyl-6-oxo-1,6-dihydropyrimidin-2-yl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine
4-(4-benzylpiperazin-1-yl)-6-methyl-2-(pyridin-3-yl)pyrimidine
5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{[(2-methoxyethyl)[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl]methyl}piperidine-4-carboxamide